Affinity DataKi: 2nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 119nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 279nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 295nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 387nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 488nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 488nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 568nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 582nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 603nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 639nMAssay Description:Displacement of [3H]ZM241383 from human A2AR expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 687nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.33E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.67E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.87E+3nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.68E+3nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.46E+3nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.54E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70E+3nMAssay Description:Displacement of [3H]DPCPX from human A1 receptor expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]AB-MEGA from human A3R expressed in CHO cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.340nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: 146nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 156nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 334nMAssay Description:Inverse agonist activity at human A2B receptor expressed in CHO cells assessed as reduction in cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human A2B receptor expressed in CHO cells assessed as reduction in cAMP productionMore data for this Ligand-Target Pair