Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50012194
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555255(CHEMBL4777388)
Affinity DataIC50:  20nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555248(CHEMBL4779439)
Affinity DataIC50:  150nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555247(CHEMBL4789394)
Affinity DataIC50:  150nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555251(CHEMBL4739952)
Affinity DataIC50:  170nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555254(CHEMBL4753496)
Affinity DataIC50:  240nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555252(CHEMBL4795173)
Affinity DataIC50:  270nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555249(CHEMBL4798520)
Affinity DataIC50:  370nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555253(CHEMBL4792301)
Affinity DataIC50:  380nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555250(CHEMBL4752826)
Affinity DataIC50:  400nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555246(CHEMBL4790861)
Affinity DataIC50:  680nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555245(CHEMBL4762047)
Affinity DataIC50:  1.50E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555236(CHEMBL4759877)
Affinity DataIC50:  1.60E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555244(CHEMBL4764244)
Affinity DataIC50:  1.80E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555239(CHEMBL4794279)
Affinity DataIC50:  2.20E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555238(CHEMBL4763642)
Affinity DataIC50:  2.40E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555240(CHEMBL4800168)
Affinity DataIC50:  2.50E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555235(CHEMBL4791418)
Affinity DataIC50:  3.70E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555234(CHEMBL4792820)
Affinity DataIC50:  4.30E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555241(CHEMBL4757746)
Affinity DataIC50:  7.40E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555237(CHEMBL4792234)
Affinity DataIC50:  7.90E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555243(CHEMBL4764592)
Affinity DataIC50:  8.00E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555242(CHEMBL4758509)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555256(CHEMBL4756115)
Affinity DataKd:  1.64E+3nMAssay Description:Binding affinity to NHERF1 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555258(CHEMBL4789294)
Affinity DataKd:  3.97E+3nMAssay Description:Binding affinity to NHERF1 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555259(CHEMBL4756359)
Affinity DataKd:  780nMAssay Description:Binding affinity to NHERF1 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555256(CHEMBL4756115)
Affinity DataKd:  1.87E+3nMAssay Description:Binding affinity to NHERF2 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555257(CHEMBL4763464)
Affinity DataKd:  560nMAssay Description:Binding affinity to NHERF2 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555258(CHEMBL4789294)
Affinity DataKd:  6.04E+3nMAssay Description:Binding affinity to NHERF2 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555259(CHEMBL4756359)
Affinity DataKd:  1.37E+3nMAssay Description:Binding affinity to NHERF2 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555256(CHEMBL4756115)
Affinity DataKd:  4.07E+3nMAssay Description:Binding affinity to NHERF2 PDZ2 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555257(CHEMBL4763464)
Affinity DataKd:  2.82E+3nMAssay Description:Binding affinity to NHERF2 PDZ2 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555258(CHEMBL4789294)
Affinity DataKd:  7.66E+3nMAssay Description:Binding affinity to NHERF2 PDZ2 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555259(CHEMBL4756359)
Affinity DataKd:  6nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence pola...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555258(CHEMBL4789294)
Affinity DataKd:  87nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence pola...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555257(CHEMBL4763464)
Affinity DataKd:  49nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence pola...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555256(CHEMBL4756115)
Affinity DataKd:  113nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence pola...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF2(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555259(CHEMBL4756359)
Affinity DataKd:  7.48E+3nMAssay Description:Binding affinity to NHERF2 PDZ2 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1(Homo sapiens)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50555257(CHEMBL4763464)
Affinity DataKd:  330nMAssay Description:Binding affinity to NHERF1 PDZ1 domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence polarization based comp...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed