Compile Data Set for Download or QSAR
maximum 50k data
Found 37 Enz. Inhib. hit(s) with all data for entry = 50013672
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50214615(CHEBI:64177 | Clobenpropit)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568499(CHEMBL4876429)
Affinity DataIC50:  2.20nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568486(CHEMBL4852639)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568492(CHEMBL4859825)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568493(CHEMBL4856094)
Affinity DataIC50:  3.40nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568494(CHEMBL4846443)
Affinity DataIC50:  4.70nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568491(CHEMBL4870117)
Affinity DataIC50:  4.90nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568500(CHEMBL4878762)
Affinity DataIC50:  5.10nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568497(CHEMBL4853496)
Affinity DataIC50:  7.10nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568485(CHEMBL4868743)
Affinity DataIC50:  8.30nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568502(CHEMBL4847024)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568501(CHEMBL4858290)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568489(CHEMBL4857779)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568495(CHEMBL4872910)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568487(CHEMBL4862604)
Affinity DataIC50:  69nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568498(CHEMBL4852674)
Affinity DataIC50:  85nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568490(CHEMBL4848375)
Affinity DataIC50:  104nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568488(CHEMBL4876778)
Affinity DataIC50:  178nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568496(CHEMBL4848524)
Affinity DataIC50:  353nMAssay Description:Antagonist activity at human H3 receptor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568499(CHEMBL4876429)
Affinity DataIC50:  2.07E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568485(CHEMBL4868743)
Affinity DataIC50:  2.24E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568494(CHEMBL4846443)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568500(CHEMBL4878762)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568486(CHEMBL4852639)
Affinity DataIC50:  3.26E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568493(CHEMBL4856094)
Affinity DataIC50:  3.29E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568489(CHEMBL4857779)
Affinity DataIC50:  3.95E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568487(CHEMBL4862604)
Affinity DataIC50:  4.12E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568490(CHEMBL4848375)
Affinity DataIC50:  4.51E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568495(CHEMBL4872910)
Affinity DataIC50:  5.32E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568497(CHEMBL4853496)
Affinity DataIC50:  5.38E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568488(CHEMBL4876778)
Affinity DataIC50:  5.54E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568496(CHEMBL4848524)
Affinity DataIC50:  6.02E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568498(CHEMBL4852674)
Affinity DataIC50:  6.18E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568492(CHEMBL4859825)
Affinity DataIC50:  6.26E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50568491(CHEMBL4870117)
Affinity DataIC50:  7.01E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50466416(CHEMBL4287929)
Affinity DataIC50:  7.12E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50:  8.27E+3nMAssay Description:Inhibition of amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs by Thioflavin T based fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed