Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 50015340
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585680BDBM50585680(CHEMBL5070349)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585682BDBM50585682(CHEMBL5085017)
Affinity DataIC50: 0.800nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585661BDBM50585661(CHEMBL5076792)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585682BDBM50585682(CHEMBL5085017)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585682BDBM50585682(CHEMBL5085017)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585678BDBM50585678(CHEMBL5093228)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585680BDBM50585680(CHEMBL5070349)
Affinity DataIC50: 1.60nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585661BDBM50585661(CHEMBL5076792)
Affinity DataIC50: 1.80nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585673BDBM50585673(CHEMBL5090020)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585661BDBM50585661(CHEMBL5076792)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585680BDBM50585680(CHEMBL5070349)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585678BDBM50585678(CHEMBL5093228)
Affinity DataIC50: 2nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585660BDBM50585660(CHEMBL5080268)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585658BDBM50585658(CHEMBL5083073)
Affinity DataIC50: 2.5nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585662BDBM50585662(CHEMBL5088686)
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585649BDBM50585649(CHEMBL5087110)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585656BDBM50585656(CHEMBL5078566)
Affinity DataIC50: 3.20nMAssay Description:Inverse agonist activity at human CB1R expressed in CHO-K1 cell membrane assessed as increase in [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585657BDBM50585657(CHEMBL5092394)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585654BDBM50585654(CHEMBL5087041)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585660BDBM50585660(CHEMBL5080268)
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585659BDBM50585659(CHEMBL5073465)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585678BDBM50585678(CHEMBL5093228)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585652BDBM50585652(CHEMBL5084492)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585658BDBM50585658(CHEMBL5083073)
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585657BDBM50585657(CHEMBL5092394)
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585683BDBM50585683(CHEMBL5071344)
Affinity DataIC50: 5.40nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585683BDBM50585683(CHEMBL5071344)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585658BDBM50585658(CHEMBL5083073)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585676BDBM50585676(CHEMBL5075684)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585673BDBM50585673(CHEMBL5090020)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585653BDBM50585653(CHEMBL5089095)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585652BDBM50585652(CHEMBL5084492)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21278BDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585668BDBM50585668(CHEMBL5081757)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585653BDBM50585653(CHEMBL5089095)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585675BDBM50585675(CHEMBL5085413)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585656BDBM50585656(CHEMBL5078566)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585671BDBM50585671(CHEMBL5084642)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585677BDBM50585677(CHEMBL5086960)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585674BDBM50585674(CHEMBL5081180)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585662BDBM50585662(CHEMBL5088686)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]- CP55940 from human CB2R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585655BDBM50585655(CHEMBL5076422)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585650BDBM50585650(CHEMBL5087924)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585654BDBM50585654(CHEMBL5087041)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585653BDBM50585653(CHEMBL5089095)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]- CP55940 from human CB2R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585667BDBM50585667(CHEMBL5086256)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585666BDBM50585666(CHEMBL5083217)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585683BDBM50585683(CHEMBL5071344)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]- CP55940 from human CB2R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21278BDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  20nMAssay Description:Antagonist activity at human CB1R expressed in CHO-K1 cell membranes assessed as stimulation of [35S]-GTPgammaS binding by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50585662BDBM50585662(CHEMBL5088686)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]- CP55940 from human CB1R expressed in CHO-K1 cells membrane by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
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