Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50002818
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024415(5-Chloro-1H-indole-2-carboxylic acid (5-imidazol-1...)
Affinity DataIC50: 7nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024424(5-Chloro-1H-indole-2-carboxylic acid (8-imidazol-1...)
Affinity DataIC50: 27nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024414(1H-Indole-2-carboxylic acid (4-imidazol-1-yl-butyl...)
Affinity DataIC50: 40nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024408(5-Chloro-1H-indole-2-carboxylic acid (3-imidazol-1...)
Affinity DataIC50: 50nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024413(5-Chloro-thiophene-2-carboxylic acid (8-imidazol-1...)
Affinity DataIC50: 70nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024412(5-Chloro-benzo[b]thiophene-2-carboxylic acid (3-im...)
Affinity DataIC50: 100nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024419(5-Chloro-thiophene-2-carboxylic acid (5-imidazol-1...)
Affinity DataIC50: 200nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024423(5-Chloro-thiophene-2-carboxylic acid (6-imidazol-1...)
Affinity DataIC50: 200nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024410(5-Chloro-thiophene-2-carboxylic acid (4-imidazol-1...)
Affinity DataIC50: 200nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024407(Benzofuran-2-carboxylic acid (3-imidazol-1-yl-prop...)
Affinity DataIC50: 300nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024420(3-Chloro-benzo[b]thiophene-2-carboxylic acid (3-im...)
Affinity DataIC50: 300nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024422(4,5-Dibromo-thiophene-2-carboxylic acid (3-imidazo...)
Affinity DataIC50: 400nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024417(5-Chloro-thiophene-2-carboxylic acid (3-imidazol-1...)
Affinity DataIC50: 600nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024418(5-Methyl-thiophene-2-carboxylic acid (3-imidazol-1...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM7962(CHEMBL537708 | 4-[2-(1H-imidazol-1-yl)ethoxy]benzo...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024409(5-Chloro-thiophene-2-carboxylic acid (3-imidazol-1...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024416(6-Chloro-N-(5-imidazol-1-yl-pentyl)-nicotinamide |...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024421(Thiophene-2-carboxylic acid (4-imidazol-1-yl-butyl...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024425(6-Chloro-N-(3-imidazol-1-yl-butyl)-nicotinamide | ...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50024411(6-Chloro-N-(4-imidazol-1-yl-butyl)-nicotinamide | ...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of thromboxane formation at a concentration of 10e -6 M.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed