Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50016963
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598700(CHEMBL5194472 | US20250084084, Example 91)
Affinity DataKi:  0.0440nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598690(CHEMBL5181223 | US20250084084, Example 1)
Affinity DataKi:  0.210nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598697(CHEMBL5179337 | US12187727, Example 64)
Affinity DataKi:  0.25nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598702(CHEMBL5173560)
Affinity DataKi:  0.280nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598703(CHEMBL5170290 | US20250084084, Example 120)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598695(CHEMBL5174952 | US20250084084, Example 6)
Affinity DataKi:  0.440nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598696(CHEMBL5183637 | US20250084084, Example 106)
Affinity DataKi:  0.460nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598699(CHEMBL5195837)
Affinity DataKi:  0.540nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598692(CHEMBL5175663 | US20250084084, Example 3)
Affinity DataKi:  0.540nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598691(CHEMBL5204022 | US20250084084, Example 2)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598693(CHEMBL5200190 | US20250084084, Example 4)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598701(CHEMBL5199107)
Affinity DataKi:  57nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598698(CHEMBL5189093)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetMelanocortin receptor 4(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50598694(CHEMBL5208472 | US20250084084, Example 5)
Affinity DataKi: >200nMAssay Description:Displacement of [125I]-[Nle4-D-phe7]-alpha-MSH from to human MC4R expressed in CHO cells incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed