Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50002882
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024694BDBM50024694((S)-6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethy...)
Affinity DataIC50: 36nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024698BDBM50024698(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024687BDBM50024687((+/-)-6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymet...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024688BDBM50024688(9-Imidazol-1-yl-8-(4-methoxy-benzyloxymethyl)-non-...)
Affinity DataIC50: 390nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024685BDBM50024685((R)-6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethy...)
Affinity DataIC50: 420nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50023002BDBM50023002(4-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 540nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024693BDBM50024693(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 560nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024684BDBM50024684(5-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 730nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024691BDBM50024691(5-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 750nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024699BDBM50024699(9-Imidazol-1-yl-8-(4-methoxy-benzyloxymethyl)-nona...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 7962BDBM7962(CHEMBL537708 | 4-[2-(1H-imidazol-1-yl)ethoxy]benzo...)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024690BDBM50024690(9-Imidazol-1-yl-8-(4-methoxy-benzyloxymethyl)-nona...)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024696BDBM50024696(7-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024686BDBM50024686(7-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024692BDBM50024692(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 8.33E+3nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024697BDBM50024697(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024695BDBM50024695(6-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane-A synthase(Human)
Searle Research and Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024689BDBM50024689(8-[2-Imidazol-1-yl-1-(4-methoxy-benzyloxymethyl)-e...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Thromboxane B2 formation in collagen-stimulated human platelets in platelet rich plasma.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed