Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 50019014
Affinity DataEC50: 14nMAssay Description:Positive allosteric modulation of mouse GPR40More data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Positive allosteric modulation of mouse GPR40More data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Positive allosteric modulation of mouse GPR40More data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 58nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 69nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Positive allosteric modulation of human GPR40 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Positive allosteric modulation of human GPR40 expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 290nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Positive allosteric modulation of human GPR40 expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 370nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 430nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 430nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 580nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 740nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 980nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Positive allosteric modulation of human GPR40 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of CYP2C8 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+3nMAssay Description:Positive allosteric modulation of human GPR40 expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+3nMAssay Description:Positive allosteric modulation of human GPR40 by calcium based FLIPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+3nMAssay Description:Positive allosteric modulation of human GPR40 expressed in HEK293 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+3nMAssay Description:Transactivation of PPARgamma (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 4.10E+3nMAssay Description:Positive allosteric modulation of human GPR40 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.30E+3nMAssay Description:Transactivation of PPARgamma (unknown origin)More data for this Ligand-Target Pair








































