Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50022333
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PARP2 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50: 8nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50650930(CHEMBL5633539)
Affinity DataIC50: 30nMAssay Description:Inhibition of PARP2 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650929(CHEMBL5634034)
Affinity DataIC50: 32nMAssay Description:Inhibition of PARP2 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650930(CHEMBL5633539)
Affinity DataIC50: 34nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650928(CHEMBL5632283)
Affinity DataIC50: 35nMAssay Description:Inhibition of PARP2 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650929(CHEMBL5634034)
Affinity DataIC50: 37nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650928(CHEMBL5632283)
Affinity DataIC50: 43nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650927(CHEMBL5632938)
Affinity DataIC50: 65nMAssay Description:Inhibition of PARP2 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650927(CHEMBL5632938)
Affinity DataIC50: 71nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650931(CHEMBL5632389)
Affinity DataIC50: 131nMAssay Description:Inhibition of PARP2 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50528813(CHEMBL4163879 | US20250101023, Example THZ531)
Affinity DataIC50: 161nMAssay Description:Inhibition of CDK12 (unknown origin) in presence of ATP by kinase-glo plus luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650931(CHEMBL5632389)
Affinity DataIC50: 167nMAssay Description:Inhibition of PARP1 (unknown origin) incubated for 1 hr by ELISA analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650931(CHEMBL5632389)
Affinity DataIC50: 269nMAssay Description:Inhibition of CDK12 (unknown origin) in presence of ATP by kinase-glo plus luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650930(CHEMBL5633539)
Affinity DataIC50: 285nMAssay Description:Inhibition of CDK12 (unknown origin) in presence of ATP by kinase-glo plus luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650929(CHEMBL5634034)
Affinity DataIC50: 344nMAssay Description:Inhibition of CDK12 (unknown origin) in presence of ATP by kinase-glo plus luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650930(CHEMBL5633539)
Affinity DataIC50: 517nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650928(CHEMBL5632283)
Affinity DataIC50: 554nMAssay Description:Inhibition of CDK12 (unknown origin) in presence of ATP by kinase-glo plus luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650930(CHEMBL5633539)
Affinity DataIC50: 689nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650930(CHEMBL5633539)
Affinity DataIC50: 748nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50650927(CHEMBL5632938)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK12 (unknown origin) in presence of ATP by kinase-glo plus luminescent assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed