Report error Found 131 Enz. Inhib. hit(s) with all data for entry = 50022355
Affinity DataKi: 5nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity to human dopamine 2 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition an...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured aft...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 26nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity to human 5HT7 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 127nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 157nMAssay Description:Binding affinity to human dopamine 2 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 169nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 169nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 178nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 178nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 179nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 179nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 181nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 187nMAssay Description:Binding affinity to human 5HT6 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 188nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 209nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 229nMAssay Description:Binding affinity to human dopamine 2 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition an...More data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Binding affinity to human dopamine 2 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 355nMAssay Description:Binding affinity to human 5HT2A receptor expressed in CHO-K1 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 362nMAssay Description:Binding affinity to human dopamine 2 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 362nMAssay Description:Binding affinity to human dopamine 2 receptor expressed in HEK293 cells assessed as inhibition constant incubated for 1 hr radioligand binding assayMore data for this Ligand-Target Pair
