Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50020297
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628622(CHEMBL5439214)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50436459(CHEMBL2396661)
Affinity DataIC50: 5nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628619(CHEMBL5422044)
Affinity DataIC50: 8.10nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628618(CHEMBL5420057)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 12nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628618(CHEMBL5420057)
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628621(CHEMBL5406498)
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628620(CHEMBL5438456)
Affinity DataIC50: 15nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628622(CHEMBL5439214)
Affinity DataIC50: 26nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628615(CHEMBL5418257)
Affinity DataIC50: 28nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 29nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628621(CHEMBL5406498)
Affinity DataIC50: 38nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628620(CHEMBL5438456)
Affinity DataIC50: 39nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628615(CHEMBL5418257)
Affinity DataIC50: 39nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628613(CHEMBL5410758)
Affinity DataIC50: 42nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628622(CHEMBL5439214)
Affinity DataIC50: 42nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628616(CHEMBL5400641)
Affinity DataIC50: 45nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628616(CHEMBL5400641)
Affinity DataIC50: 48nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628619(CHEMBL5422044)
Affinity DataIC50: 53nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628614(CHEMBL5435973)
Affinity DataIC50: 56nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50436459(CHEMBL2396661)
Affinity DataIC50: 69nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50436459(CHEMBL2396661)
Affinity DataIC50: 102nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628617(CHEMBL5410409)
Affinity DataIC50: 130nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628617(CHEMBL5410409)
Affinity DataIC50: 140nMAssay Description:Inhibition of PI3K alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628613(CHEMBL5410758)
Affinity DataIC50: 152nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 11(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50188961(CHEMBL3622533)
Affinity DataIC50: 177nMAssay Description:Inhibition of HDAC11 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628618(CHEMBL5420057)
Affinity DataIC50: 214nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628622(CHEMBL5439214)
Affinity DataIC50: 285nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628618(CHEMBL5420057)
Affinity DataIC50: 318nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628618(CHEMBL5420057)
Affinity DataIC50: 471nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 11(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628622(CHEMBL5439214)
Affinity DataIC50: 586nMAssay Description:Inhibition of HDAC11 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 6(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628614(CHEMBL5435973)
Affinity DataIC50: 680nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 814nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628622(CHEMBL5439214)
Affinity DataIC50: 880nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50436459(CHEMBL2396661)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628618(CHEMBL5420057)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 11(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628618(CHEMBL5420057)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HDAC11 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628622(CHEMBL5439214)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 8(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628618(CHEMBL5420057)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandPNGBDBM50628622(CHEMBL5439214)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed