Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50021236
Affinity DataKi: 0.200nMAssay Description:Binding affinity to human TRPV1 expressed in HEK293 cells assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of heat shock (45 degreeC)-induced increase in intracellular Ca2+...More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of capsaicin-induced increase in Ca2+ fluxMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ level by FLIP...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ level by FLIP...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at rat TRPV1 assessed as inhibition of pH-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at rat TRPV1 assessed as inhibition of pH-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of pH-induced increase in intracellular Ca2+ level by calcium flu...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of NADA-induced increase in intracellular Ca2+ level incubated fo...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Antagonist activity at rat TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ level by FLIPR-...More data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ level by FLIP...More data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:Antagonist activity at capsaicin-induced human TRPV1 activationMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human TRPV1More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of COX-2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ level incubat...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced Ca2+ influx by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of COX-2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity to MOR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity to human TRPV1 assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Antagonist activity at rat TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ level by FLIPR-...More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of rat TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of rat TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of pH-induced increase in intracellular Ca2+ level by fluorescence bas...More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of 5-LOX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 313nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of pH-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Inhibition of 5-LOX (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of resiniferatoxin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 2.39E+3nMAssay Description:Antagonist activity at rat TRPA1 assessed as inhibition of AITC-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 8.64E+3nMAssay Description:Antagonist activity at rat TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+4nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of AITC-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+4nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ levelMore data for this Ligand-Target Pair
