Report error Found 126 Enz. Inhib. hit(s) with all data for entry = 50021529
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 0.120nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 0.240nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Binding affinity to PIM2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataKi: 0.550nMAssay Description:Binding affinity to PIM1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of PIM3 (unknown origin) by FRET based Z-LYTE kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human full length-His6 tagged PIM1 (1 to 312 residues) expressed in Escherichia coli BL21 (DE3) using RSRHSSYPAGT as peptide substrate ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human PIM1 using KKRNRTLTK as substrate in presence of [gamma-33P]-ATP by hotspot kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of PIM3 (unknown origin) by FRET based Z-LYTE kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of PIM2 (unknown origin) by FRET based Z-LYTE kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of human full length-His6 tagged PIM1 (1 to 312 residues) expressed in Escherichia coli BL21 (DE3) using RSRHSSYPAGT as peptide substrate ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of PIM2 (unknown origin) by FRET based Z-LYTE kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 9.30nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of PIM2 (unknown origin) by FRET based Z-LYTE kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of PIM3 (unknown origin) by FRET based Z-LYTE kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human PIM1 by discoverX kinome scan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human PIM1 by discoverX kinome scan assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of CLK1 (unknown origin) using GRSRSRSRSRSRSRS as substrate incubated for 15 mins in presence of ATP by gamma32P-ATP based analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of COX2 (unknown origin) fluorescence based analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of human full length-His6 tagged PIM2 (1 to 311 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using R...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of PIM2 (unknown origin) by FRET based Z-LYTE kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of human PIM1 by discoverX kinome scan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human PIM2 by ADP-Glo luminescent assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human PIM1 by ADP Glo luminescent assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human PIM1 by discoverX kinome scan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of PIM3 (unknown origin) by FRET based Z-LYTE kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of human PIM1 by discoverX kinome scan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Human)
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Joint Research Institution of Altitude Health and Institute of Respiratory Health and National Clinical Research Center for Geriatrics
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of COX2 (unknown origin) fluorescence based analysisMore data for this Ligand-Target Pair






3D Structure (crystal)
























