Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50021017
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50511906(CHEMBL4435830 | US11045448, Cpd. No. 57)
Affinity DataIC50: 3.30nMAssay Description:Binding affinity to menin (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636089(CHEMBL5565919)
Affinity DataIC50: 250nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636083(CHEMBL5527907)
Affinity DataIC50: 380nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636085(CHEMBL5555656)
Affinity DataIC50: 450nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636086(CHEMBL5557085)
Affinity DataIC50: 470nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636087(CHEMBL5557705)
Affinity DataIC50: 530nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM152235(US8993552, 70)
Affinity DataIC50: 600nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636084(CHEMBL5518084)
Affinity DataIC50: 730nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636088(CHEMBL5560342)
Affinity DataIC50: 1.04E+3nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636091(CHEMBL5562800)
Affinity DataIC50: 1.14E+3nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636090(CHEMBL5559575)
Affinity DataIC50: 1.22E+3nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636078(CHEMBL5558500)
Affinity DataIC50: 1.47E+3nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636080(CHEMBL5560540)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636079(CHEMBL5557241)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636082(CHEMBL5566849)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMenin(Human)
Xi'an Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50636081(CHEMBL5532611)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to menin (unknown origin) incubated for 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed