Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50021056
TargetHistone acetyltransferase p300(Human)
Guangzhou Institutes of Biomedicine and Health
Curated by ChEMBL
Guangzhou Institutes of Biomedicine and Health
Curated by ChEMBL
Affinity DataKd: 1.30nMAssay Description:Binding affinity to p300 (unknown origin) by SPR methodMore data for this Ligand-Target Pair
Affinity DataKd: 1.70nMAssay Description:Binding affinity to CBP (unknown origin) by SPR methodMore data for this Ligand-Target Pair
Affinity DataKd: 21nMAssay Description:Binding affinity to human CBP by ITC methodMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Human)
Guangzhou Institutes of Biomedicine and Health
Curated by ChEMBL
Guangzhou Institutes of Biomedicine and Health
Curated by ChEMBL
Affinity DataKd: 32nMAssay Description:Binding affinity to human p300 by ITC methodMore data for this Ligand-Target Pair
Affinity DataIC50: 91nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 134nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 166nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 214nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 257nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 444nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 484nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+3nMAssay Description:Binding affinity to CBP BD (unknown origin) incubated for 2.5 hrs by Alphascreen assayMore data for this Ligand-Target Pair









