Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50021344
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  24nMAssay Description:Agonist activity against rat mGlu4 K74A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50639733(CHEMBL5561878)
Affinity DataIC50: 80nMAssay Description:Inhibition of [3H] -LY341495 binding to rat mGlu7 expressed in CHO cell membrane incubated for 30 mins in presence of LY341495 by liquid scintillatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50062522((1S,2S)-2-[(1S)-1-amino-1-carboxy-2-(9H-xanthen-9-...)
Affinity DataIC50: 190nMAssay Description:Inhibition of [3H] -LY341495 binding to rat mGlu7 expressed in CHO cell membrane incubated for 30 mins by liquid scintillation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50007548(2-Amino-4-phosphono-butyric acid | 2-amino-4-phosp...)
Affinity DataEC50:  230nMAssay Description:Agonist activity against rat mGlu4 K74A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50007548(2-Amino-4-phosphono-butyric acid | 2-amino-4-phosp...)
Affinity DataEC50:  1.16E+3nMAssay Description:Agonist activity against rat mGlu4 R60A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50007548(2-Amino-4-phosphono-butyric acid | 2-amino-4-phosp...)
Affinity DataEC50:  1.87E+3nMAssay Description:Agonist activity at rat mGlu4 R258A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50007548(2-Amino-4-phosphono-butyric acid | 2-amino-4-phosp...)
Affinity DataEC50:  2.66E+3nMAssay Description:Agonist activity against rat mGlu4 S160A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  4.91E+3nMAssay Description:Agonist activity at rat mGlu4 R258A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  9.07E+3nMAssay Description:Agonist activity against rat mGlu4 R60A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50007548(2-Amino-4-phosphono-butyric acid | 2-amino-4-phosp...)
Affinity DataEC50:  1.05E+4nMAssay Description:Agonist activity at rat mGlu7 N74K mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50007548(2-Amino-4-phosphono-butyric acid | 2-amino-4-phosp...)
Affinity DataEC50:  1.23E+4nMAssay Description:Agonist activity against rat mGlu4 S160D mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  1.82E+4nMAssay Description:Agonist activity at rat mGlu7 Q258A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  1.85E+4nMAssay Description:Agonist activity against rat mGlu4 S160D mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 4(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  2.62E+4nMAssay Description:Agonist activity against rat mGlu4 S160A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  3.20E+4nMAssay Description:Agonist activity at rat mGlu7 N74A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  4.70E+4nMAssay Description:Agonist activity at rat mGlu7 N74K mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50007548(2-Amino-4-phosphono-butyric acid | 2-amino-4-phosp...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat mGlu7 N74A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50:  1.78E+5nMAssay Description:Agonist activity at rat mGlu7 K60A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50: >3.00E+5nMAssay Description:Agonist activity at rat mGlu7 K60A/S160A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM196906(US9212196, Derivative 2)
Affinity DataEC50: >3.00E+5nMAssay Description:Agonist activity at rat mGlu7 S160A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMetabotropic glutamate receptor 7(Rat)
Universite Paris Cite

Curated by ChEMBL
LigandPNGBDBM50007548(2-Amino-4-phosphono-butyric acid | 2-amino-4-phosp...)
Affinity DataEC50:  1.98E+6nMAssay Description:Agonist activity at rat mGlu7 K60A mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed