Affinity DataIC50: 23nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of human kidney microsomal COX assessed as PGE2 level using arachidonic acid as substrate preincubated for 5 to 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of human kidney microsomal COX assessed as PGE2 level using arachidonic acid as substrate preincubated for 5 to 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of human kidney microsomal COX assessed as PGE2 level using arachidonic acid as substrate preincubated for 5 to 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition concentration against human adenosine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Compound was evaluated for its binding affinity against Toxoplasma gondii purine nucleoside phosphorylase of virulent strain RH (value indicates comp...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Inhibition of human kidney microsomal COX assessed as PGE2 level using arachidonic acid as substrate preincubated for 5 to 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Inhibition concentration against human adenosine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 104nMAssay Description:Inhibition of rat kidney microsomal COX assessed as PGE2 level using arachidonic acid as substrate preincubated for 5 to 15 mins followed by substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Inhibition of rat kidney microsomal COX assessed as PGE2 level using arachidonic acid as substrate preincubated for 5 to 15 mins followed by substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 128nMAssay Description:Inhibition of rat kidney microsomal COX assessed as PGE2 level using arachidonic acid as substrate preincubated for 5 to 15 mins followed by substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 132nMAssay Description:Inhibition of rat kidney microsomal COX assessed as PGE2 level using arachidonic acid as substrate preincubated for 5 to 15 mins followed by substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 132nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 141nMAssay Description:Binding affinity towards Alpha-1A adrenergic receptor in rat denuded thoracic aortaMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of human COX-2 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 45 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of Platelet-derived growth factor receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of human COX-2 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 45 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human COX-2 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 45 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Antagonistic activity at human progesterone receptor in CV-1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:Inhibition of human COX-2 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 45 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 790nMAssay Description:Inhibition of human COX-2 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 45 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 810nMAssay Description:Inhibition concentration against human adenosine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 880nMAssay Description:Inhibition of human COX-2 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 45 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 910nMAssay Description:Binding affinity to human progesterone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 970nMAssay Description:Inhibition of Dexamethasone stimulated transcriptional activity in CHO cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of human COX-2 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 45 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human COX-1 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by t...More data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+5nMAssay Description:Inhibition of human COX-1 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by t...More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+5nMAssay Description:Inhibition of human COX-1 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by t...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of human COX-1 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by t...More data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+5nMAssay Description:Inhibition of human COX-1 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by t...More data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of human COX-1 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by t...More data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+5nMAssay Description:Antiviral activity against human rhinovirus-14 (HRV-14) 3C protease using enzyme assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.67E+5nMAssay Description:Inhibition concentration against human adenosine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.78E+5nMAssay Description:Inhibition of human COX-1 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by t...More data for this Ligand-Target Pair
Affinity DataIC50: 2.01E+5nMAssay Description:Inhibition of human COX-1 using [14C]-arachidonic acid as substrate preincubated for 5 mins followed by substrate addition measured after 2 mins by t...More data for this Ligand-Target Pair