Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50012318
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556491(CHEMBL4784458)
Affinity DataIC50:  6.74E+3nMAssay Description:Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556492(CHEMBL4747352)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556488(CHEMBL4756022)
Affinity DataKd:  890nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556489(CHEMBL4755703)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556490(CHEMBL4748826)
Affinity DataKd:  670nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556491(CHEMBL4784458)
Affinity DataKd:  370nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556492(CHEMBL4747352)
Affinity DataKd:  185nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556493(CHEMBL3561645)
Affinity DataKd:  3.50E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556494(CHEMBL4754833)
Affinity DataKd:  4.90E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556495(CHEMBL4796843)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556496(CHEMBL4776753)
Affinity DataKd:  8.20E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556487(CHEMBL4763249)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556488(CHEMBL4756022)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556491(CHEMBL4784458)
Affinity DataKd:  6.30E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556492(CHEMBL4747352)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556487(CHEMBL4763249)
Affinity DataKd:  400nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50556486(CHEMBL1508421)
Affinity DataKd:  1.40E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada

Curated by ChEMBL
LigandPNGBDBM50342854(1-Benzyl-4-(pyrrolidin-1-yl)pyridinium Bromide | C...)
Affinity DataKd:  2.40E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed