Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50012521
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50424917BDBM50424917(CHEMBL2311578)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 100 uM ATP as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558084BDBM50558084(CHEMBL4799933)
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 100 uM ATP as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558084BDBM50558084(CHEMBL4799933)
Affinity DataKi:  740nMAssay Description:Uncompetitive inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558079BDBM50558079(CHEMBL4795698)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558084BDBM50558084(CHEMBL4799933)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558084BDBM50558084(CHEMBL4799933)
Affinity DataKi:  3.50E+3nMAssay Description:Competitive inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558068BDBM50558068(CHEMBL4744813)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 100 uM ATP as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558080BDBM50558080(CHEMBL4796698)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558068BDBM50558068(CHEMBL4744813)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558087BDBM50558087(CHEMBL4791393)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 100 uM ATP as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558074BDBM50558074(CHEMBL4756969)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558078BDBM50558078(CHEMBL4742336)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558076BDBM50558076(CHEMBL4749702)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558068BDBM50558068(CHEMBL4744813)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 5 uM ATP as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558072BDBM50558072(CHEMBL4763020)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558075BDBM50558075(CHEMBL4751086)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558077BDBM50558077(CHEMBL4741172)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558081BDBM50558081(CHEMBL4764224)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50526600BDBM50526600(CHEMBL4584982)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558082BDBM50558082(CHEMBL4776652)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558083BDBM50558083(CHEMBL4776353)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558069BDBM50558069(CHEMBL4755450)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558085BDBM50558085(CHEMBL4750198)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558070BDBM50558070(CHEMBL4747454)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558071BDBM50558071(CHEMBL4752647)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558086BDBM50558086(CHEMBL4746514)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 100 uM ATP as subst...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTransitional endoplasmic reticulum ATPase(Human)
University of Pittsburgh

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50558073BDBM50558073(CHEMBL4792968)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human full length Avi-tagged p97 (1 to 806 residues) expressed in Escherichia coli Rosetta 2(DE3) using 20 uM ATP as substr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed