Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
Affinity DataIC50: 2.86E+5nMAssay Description:Inhibition of COX-2 (unknown origin) using arachidonic acid as substrate preincubated for 10 mins followed by substrate addition by microplate reader...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 1.84E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 6.41E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 1.18E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 930nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 4.61E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 1.74E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 6.29E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 5.30E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 1.20E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 5.25E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 7.94E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 6.67E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 2.47E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 1.73E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 960nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 1.71E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 1.22E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 5.52E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 2.46E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 4.00E+3nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: 2.16E+4nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to GAL4-DBD-fused PPARgamma ligand binding domain (unknown origin) expressed in HEK293T cells by spectra-fluorophotometry analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 1.17E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 2.27E+4nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Xiamen University
Curated by ChEMBL
Xiamen University
Curated by ChEMBL
Affinity DataEC50: 2.78E+3nMAssay Description:Partial agonist activity at GAL4 DBD-fused PPARgamma LBD (unknown origin) expressed in pG5 luc and pBIND transfected HEK293T cells assessed as transc...More data for this Ligand-Target Pair