Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50015561
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522280BDBM522280(US11161839, Example 10a)
Affinity DataIC50: 3nMAssay Description:Inhibition of BCOR peptide binding to human BCL6 expressed in Escherichia coli measured after 270 mins by BCOR ULight TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522280BDBM522280(US11161839, Example 10a)
Affinity DataIC50: 26nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522280BDBM522280(US11161839, Example 10a)
Affinity DataIC50: 26nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50546197BDBM50546197(CHEMBL4755229)
Affinity DataIC50: 30nMAssay Description:Inhibition of BCOR peptide binding to human BCL6 expressed in Escherichia coli measured after 270 mins by BCOR ULight TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587565BDBM50587565(CHEMBL5081226)
Affinity DataIC50: 46nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522284BDBM522284(US11161839, Example 10e)
Affinity DataIC50: 54nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522285BDBM522285(US11161839, Example 10f)
Affinity DataIC50: 73nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522286BDBM522286(US11161839, Example 10g)
Affinity DataIC50: 82nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522196BDBM522196(US11161839, Example 1b | US11161839, Example 1a)
Affinity DataIC50: 140nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522291BDBM522291(US11161839, Example 10l)
Affinity DataIC50: 200nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522280BDBM522280(US11161839, Example 10a)
Affinity DataKd:  234nMAssay Description:Binding affinity to human BCL6 BDB domain by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522235BDBM522235(US11161839, Example 3p)
Affinity DataIC50: 250nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522312BDBM522312(US11161839, Example 11i)
Affinity DataIC50: 320nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522274BDBM522274(US11161839, Example 9l)
Affinity DataIC50: 350nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522311BDBM522311(US11161839, Example 11h)
Affinity DataIC50: 420nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587565BDBM50587565(CHEMBL5081226)
Affinity DataIC50: 470nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587560BDBM50587560(CHEMBL5079024)
Affinity DataIC50: 550nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522280BDBM522280(US11161839, Example 10a)
Affinity DataIC50: 570nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587564BDBM50587564(CHEMBL5089812)
Affinity DataIC50: 790nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522227BDBM522227(US11161839, Example 3l)
Affinity DataIC50: 870nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522266BDBM522266(US11161839, Example 9c)
Affinity DataIC50: 880nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522237BDBM522237(US11161839, Example 4)
Affinity DataIC50: 900nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522226BDBM522226(US11161839, Example 1p)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587562BDBM50587562(CHEMBL5076223)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522285BDBM522285(US11161839, Example 10f)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522284BDBM522284(US11161839, Example 10e)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587554BDBM50587554(CHEMBL5090262)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522196BDBM522196(US11161839, Example 1b | US11161839, Example 1a)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587558BDBM50587558(CHEMBL5079963)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587559BDBM50587559(CHEMBL5088786)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587557BDBM50587557(CHEMBL5080619)
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522312BDBM522312(US11161839, Example 11i)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587556BDBM50587556(CHEMBL5080184)
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587555BDBM50587555(CHEMBL5090408)
Affinity DataIC50: 2.64E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587561BDBM50587561(CHEMBL5075468)
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587552BDBM50587552(CHEMBL5084602)
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 522311BDBM522311(US11161839, Example 11h)
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of human nanoLuc-tagged BCL6 expressed in HEK293T cells coexpressing HaloTag-SMRT using NanoBRET furimazine substrate incubated for 6 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587553BDBM50587553(CHEMBL5081011)
Affinity DataIC50: 5.57E+3nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMed
TargetB-cell lymphoma 6 protein(Human)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50587563BDBM50587563(CHEMBL5080163)
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of human BCL6 (5 to 129 residues) expressed in Escherichia coli BL21-AI using BCOR-AF633 peptide as substrate measured after 2 hrs by TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)