Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50029137
TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019191BDBM50019191(CHEMBL71079 | 1-Methyl-1H-indole-2-carboxylic acid...)
Affinity DataIC50: 1.40nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281711BDBM50281711(1-(4-Chloro-phenyl)-3-((R)-1-methyl-2-oxo-5-phenyl...)
Affinity DataIC50: 5.5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019240BDBM50019240(CHEMBL72073 | 4-Chloro-N-(1-methyl-2-oxo-5-phenyl-...)
Affinity DataIC50: 8.30nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281711BDBM50281711(1-(4-Chloro-phenyl)-3-((R)-1-methyl-2-oxo-5-phenyl...)
Affinity DataIC50: 12nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281703BDBM50281703(N-(9H-beta-Carbolin-3-yl)-2-(1H-indol-3-yl)-acetam...)
Affinity DataIC50: 24nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281701BDBM50281701(1-(4-Chloro-phenyl)-3-((S)-1-methyl-2-oxo-5-phenyl...)
Affinity DataIC50: 26nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281712BDBM50281712(N-(9H-beta-Carbolin-3-yl)-2-phenyl-acetamide | CHE...)
Affinity DataIC50: 40nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281705BDBM50281705(1-(9H-beta-Carbolin-3-yl)-3-(4-chloro-phenyl)-urea...)
Affinity DataIC50: 85nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281707BDBM50281707(1-(9H-beta-Carbolin-3-yl)-3-((R)-1-methyl-2-oxo-5-...)
Affinity DataIC50: 89nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281713BDBM50281713(1-(9H-beta-Carbolin-3-yl)-3-((S)-1-methyl-2-oxo-5-...)
Affinity DataIC50: 110nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281707BDBM50281707(1-(9H-beta-Carbolin-3-yl)-3-((R)-1-methyl-2-oxo-5-...)
Affinity DataIC50: 270nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281704BDBM50281704(N-(9H-beta-Carbolin-3-yl)-3-phenyl-propionamide | ...)
Affinity DataIC50: 330nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281707BDBM50281707(1-(9H-beta-Carbolin-3-yl)-3-((R)-1-methyl-2-oxo-5-...)
Affinity DataIC50: 400nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281701BDBM50281701(1-(4-Chloro-phenyl)-3-((S)-1-methyl-2-oxo-5-phenyl...)
Affinity DataIC50: 410nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281701BDBM50281701(1-(4-Chloro-phenyl)-3-((S)-1-methyl-2-oxo-5-phenyl...)
Affinity DataIC50: 540nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281709BDBM50281709(1-Methyl-1H-indole-2-carboxylic acid (9H-beta-carb...)
Affinity DataIC50: 710nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281706BDBM50281706(2-(1H-Indol-3-yl)-N-(1-methyl-2-oxo-5-phenyl-2,3-d...)
Affinity DataIC50: 1.00E+3nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281711BDBM50281711(1-(4-Chloro-phenyl)-3-((R)-1-methyl-2-oxo-5-phenyl...)
Affinity DataIC50: 1.10E+3nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50019191BDBM50019191(CHEMBL71079 | 1-Methyl-1H-indole-2-carboxylic acid...)
Affinity DataIC50: 2.00E+3nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281702BDBM50281702(N-(9H-beta-Carbolin-3-yl)-4-chloro-benzamide | CHE...)
Affinity DataIC50: 3.50E+3nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281713BDBM50281713(1-(9H-beta-Carbolin-3-yl)-3-((S)-1-methyl-2-oxo-5-...)
Affinity DataIC50: 5.90E+3nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50019240BDBM50019240(CHEMBL72073 | 4-Chloro-N-(1-methyl-2-oxo-5-phenyl-...)
Affinity DataIC50: 6.70E+3nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281714BDBM50281714(N-(9H-beta-Carbolin-3-yl)-benzamide | CHEMBL171940)
Affinity DataIC50: 7.10E+3nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281713BDBM50281713(1-(9H-beta-Carbolin-3-yl)-3-((S)-1-methyl-2-oxo-5-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281706BDBM50281706(2-(1H-Indol-3-yl)-N-(1-methyl-2-oxo-5-phenyl-2,3-d...)
Affinity DataIC50: 1.10E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281712BDBM50281712(N-(9H-beta-Carbolin-3-yl)-2-phenyl-acetamide | CHE...)
Affinity DataIC50: 1.40E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50019191BDBM50019191(CHEMBL71079 | 1-Methyl-1H-indole-2-carboxylic acid...)
Affinity DataIC50: 1.50E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281706BDBM50281706(2-(1H-Indol-3-yl)-N-(1-methyl-2-oxo-5-phenyl-2,3-d...)
Affinity DataIC50: 3.20E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281712BDBM50281712(N-(9H-beta-Carbolin-3-yl)-2-phenyl-acetamide | CHE...)
Affinity DataIC50: 3.40E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281704BDBM50281704(N-(9H-beta-Carbolin-3-yl)-3-phenyl-propionamide | ...)
Affinity DataIC50: 3.50E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50019240BDBM50019240(CHEMBL72073 | 4-Chloro-N-(1-methyl-2-oxo-5-phenyl-...)
Affinity DataIC50: 4.00E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281703BDBM50281703(N-(9H-beta-Carbolin-3-yl)-2-(1H-indol-3-yl)-acetam...)
Affinity DataIC50: 6.70E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281704BDBM50281704(N-(9H-beta-Carbolin-3-yl)-3-phenyl-propionamide | ...)
Affinity DataIC50: 6.80E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281702BDBM50281702(N-(9H-beta-Carbolin-3-yl)-4-chloro-benzamide | CHE...)
Affinity DataIC50: 7.20E+4nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001472BDBM50001472(CHEMBL54381 | 9H-beta-Carbolin-3-ylamine)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281705BDBM50281705(1-(9H-beta-Carbolin-3-yl)-3-(4-chloro-phenyl)-urea...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281702BDBM50281702(N-(9H-beta-Carbolin-3-yl)-4-chloro-benzamide | CHE...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281708BDBM50281708((S)-3-Amino-1-methyl-5-phenyl-1,3-dihydro-benzo[e]...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281705BDBM50281705(1-(9H-beta-Carbolin-3-yl)-3-(4-chloro-phenyl)-urea...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281714BDBM50281714(N-(9H-beta-Carbolin-3-yl)-benzamide | CHEMBL171940)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50243981BDBM50243981(CHEMBL453066 | Beta CCM | Methyl Beta-carboline-3 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50243981BDBM50243981(CHEMBL453066 | Beta CCM | Methyl Beta-carboline-3 ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50001472BDBM50001472(CHEMBL54381 | 9H-beta-Carbolin-3-ylamine)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281710BDBM50281710((R)-3-Amino-1-methyl-5-phenyl-1,3-dihydro-benzo[e]...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281709BDBM50281709(1-Methyl-1H-indole-2-carboxylic acid (9H-beta-carb...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281710BDBM50281710((R)-3-Amino-1-methyl-5-phenyl-1,3-dihydro-benzo[e]...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50281710BDBM50281710((R)-3-Amino-1-methyl-5-phenyl-1,3-dihydro-benzo[e]...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50001472BDBM50001472(CHEMBL54381 | 9H-beta-Carbolin-3-ylamine)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281708BDBM50281708((S)-3-Amino-1-methyl-5-phenyl-1,3-dihydro-benzo[e]...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]CCK-33 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50281703BDBM50281703(N-(9H-beta-Carbolin-3-yl)-2-(1H-indol-3-yl)-acetam...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for its activity to inhibit the binding of [125I]gastrin to gastric glands (gastrin) in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

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