Affinity DataIC50: 2nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin A recep...More data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin A recep...More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin B recep...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of sarafotoxin-6c stimulated vasoconstriction in rabbit pulmonary artery.More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin B recep...More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of sarafotoxin-6c stimulated vasoconstriction in rabbit pulmonary artery.More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin A recep...More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin A recep...More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 740nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin B recep...More data for this Ligand-Target Pair
Affinity DataIC50: 760nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin B recep...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of ET- 1 stimulated arachidonic acid release (AAR) in cultured rabbit renal vascular smooth muscle cells expressing the endothelin A recep...More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Affinity for human endothelin A receptor expressed in Ltk cells.More data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Compound was evaluated for the receptor binding activity in rabbit artery vascular smooth muscle cells expressing Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Compound was evaluated for the receptor binding activity in rabbit artery vascular smooth muscle cells expressing Endothelin A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 7.40E+3nMAssay Description:Affinity for human endothelin B receptor expressed in CHO-K1 cells.More data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of sarafotoxin-6c stimulated vasoconstriction in rabbit pulmonary artery.More data for this Ligand-Target Pair