Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50029930
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50228840((S)-1-[(R)-2-(3,3-dimethyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory concentration of the compound against trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289436((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50:  6.40nMAssay Description:Inhibitory concentration of the compound against trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289436((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration of the compound against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289434((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50: <25nMAssay Description:Inhibitory concentration against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289434((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50:  25nMAssay Description:Inhibitory concentration of the compound against trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50228840((S)-1-[(R)-2-(3,3-dimethyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50:  68nMAssay Description:Inhibitory concentration of the compound against thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289435((S)-1-[(R)-2-(3,3-Dimethyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50:  92nMAssay Description:Inhibitory concentration of the compound against thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289433((S)-1-((R)-2-Acetylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50:  156nMAssay Description:Inhibitory concentration of the compound against trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289433((S)-1-((R)-2-Acetylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50:  284nMAssay Description:Inhibitory concentration of the compound against thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289435((S)-1-[(R)-2-(3,3-Dimethyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50:  1.01E+3nMAssay Description:Inhibitory concentration of the compound against trypsin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50228840((S)-1-[(R)-2-(3,3-dimethyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibitory concentration of the compound against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289433((S)-1-((R)-2-Acetylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibitory concentration of the compound against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289434((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibitory concentration of the compound against thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289436((S)-2-((R)-2-Acetylamino-3-phenyl-propionylamino)-...)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibitory concentration of the compound against thrombin(FIIa).More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlasminogen(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289435((S)-1-[(R)-2-(3,3-Dimethyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibitory concentration of the compound against plasmin.More data for this Ligand-Target Pair
In DepthDetails Article