Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50030057
TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290697({2-[3-(3-Carbamimidoyl-phenyl)-5-(4-carbamimidoyl-...)
Affinity DataKi:  18nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM17283((2S)-3-(7-carbamimidoylnaphthalen-2-yl)-2-(4-{[(3S...)
Affinity DataKi:  41nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  94nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290699([3-(4-Carbamimidoyl-phenyl)-5-(3-carbamimidoyl-phe...)
Affinity DataKi:  117nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290692([3-(3-Carbamimidoyl-phenyl)-5-(4-carbamimidoyl-phe...)
Affinity DataKi:  143nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290690([3-(3-Carbamimidoyl-phenyl)-5-(3-carbamimidoyl-phe...)
Affinity DataKi:  230nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290694(3-(3-Carbamimidoyl-phenyl)-4,5-dihydro-isoxazole-5...)
Affinity DataKi:  270nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290697({2-[3-(3-Carbamimidoyl-phenyl)-5-(4-carbamimidoyl-...)
Affinity DataKi:  420nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  480nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290693(N-(3-Carbamimidoyl-phenyl)-2-[3-(4-carbamimidoyl-p...)
Affinity DataKi:  510nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290694(3-(3-Carbamimidoyl-phenyl)-4,5-dihydro-isoxazole-5...)
Affinity DataKi:  700nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290690([3-(3-Carbamimidoyl-phenyl)-5-(3-carbamimidoyl-phe...)
Affinity DataKi:  800nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290693(N-(3-Carbamimidoyl-phenyl)-2-[3-(4-carbamimidoyl-p...)
Affinity DataKi:  870nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290692([3-(3-Carbamimidoyl-phenyl)-5-(4-carbamimidoyl-phe...)
Affinity DataKi: >1.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290699([3-(4-Carbamimidoyl-phenyl)-5-(3-carbamimidoyl-phe...)
Affinity DataKi: >1.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetSerine protease 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290695(N-(3-Carbamimidoyl-phenyl)-2-[3-(3-carbamimidoyl-p...)
Affinity DataKi: >1.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290691(N-(4-Carbamimidoyl-phenyl)-2-[3-(3-carbamimidoyl-p...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290698(N-(4-Carbamimidoyl-phenyl)-2-[3-(4-carbamimidoyl-p...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290695(N-(3-Carbamimidoyl-phenyl)-2-[3-(3-carbamimidoyl-p...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290698(N-(4-Carbamimidoyl-phenyl)-2-[3-(4-carbamimidoyl-p...)
Affinity DataKi:  2.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290693(N-(3-Carbamimidoyl-phenyl)-2-[3-(4-carbamimidoyl-p...)
Affinity DataKi:  2.20E+3nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290697({2-[3-(3-Carbamimidoyl-phenyl)-5-(4-carbamimidoyl-...)
Affinity DataKi:  3.10E+3nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290691(N-(4-Carbamimidoyl-phenyl)-2-[3-(3-carbamimidoyl-p...)
Affinity DataKi:  1.11E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290695(N-(3-Carbamimidoyl-phenyl)-2-[3-(3-carbamimidoyl-p...)
Affinity DataKi:  1.12E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290690([3-(3-Carbamimidoyl-phenyl)-5-(3-carbamimidoyl-phe...)
Affinity DataKi:  1.18E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50066615(2-[1-[4-amino(imino)methylphenyl]-(E)-methylidene]...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290699([3-(4-Carbamimidoyl-phenyl)-5-(3-carbamimidoyl-phe...)
Affinity DataKi:  1.41E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  1.60E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290694(3-(3-Carbamimidoyl-phenyl)-4,5-dihydro-isoxazole-5...)
Affinity DataKi:  1.60E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetProthrombin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290692([3-(3-Carbamimidoyl-phenyl)-5-(4-carbamimidoyl-phe...)
Affinity DataKi: >2.10E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50058875(CHEMBL293610 | CHEMBL97570 | (S)-3-{2-[3-(4-Carbam...)
Affinity DataKi:  3.85E+4nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCoagulation factor X(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50041220(1,2-bis(5-amidinobenzofuran-2-yl)ethane | 2-(2-{5-...)
Affinity DataKi:  5.70E+5nMAssay Description:The compound was evaluated for inhibitory activity against bovine Factor XaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article