Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50034705
TargetTubulin alpha-1A chain(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50139772(leurocristine | 22-oxovincaleukoblastine | vincris...)
Affinity DataIC50: 220nMAssay Description:The compound was evaluated in vitro for the mammalian brain tubulin polymerization using standard assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

TargetTubulin alpha-1A chain(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50280140([6-(3,4,5-Trimethoxy-benzyloxy)-imidazo[1,2-b]pyri...)
Affinity DataIC50: 310nMAssay Description:In vitro mammalian brain tubulin polymerization using standard assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

TargetTubulin alpha-1A chain(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50280140([6-(3,4,5-Trimethoxy-benzyloxy)-imidazo[1,2-b]pyri...)
Affinity DataKi:  750nMAssay Description:Compound was tested for competitive inhibition with radioligand [3H]colchicine at colchicine site of mammalian tubulinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

TargetTubulin alpha-1A chain(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50014846(7alphaH-colchicine | (S)-N-(5,6,7,9-tetrahydro-1,2...)
Affinity DataIC50: 1.50E+3nMAssay Description:The compound was evaluated in vitro for the mammalian brain tubulin polymerization using standard assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article