Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50034802
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50326659(3,10-dimethoxy-17-methyl-(10S)-17-azatetracyclo[7....)
Affinity DataKi:  0.700nMAssay Description:Binding affinity by its ability to displace [3H]DAMGO from mu receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50285003(3,10-dimethoxy-17-phenethyl-17-azatetracyclo[7.5.3...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity by its ability to displace [3H]DAMGO from mu receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50326659(3,10-dimethoxy-17-methyl-(10S)-17-azatetracyclo[7....)
Affinity DataKi:  1.5nMAssay Description:Binding affinity by its ability to displace [3H]-U-69,593 from kappa receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50148071((-)-N-(Cycloproylmethyl)-4,14-dimethoxymorphinan-6...)
Affinity DataKi:  24nMAssay Description:Binding affinity by its ability to displace [3H]DAMGO from mu receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50326659(3,10-dimethoxy-17-methyl-(10S)-17-azatetracyclo[7....)
Affinity DataKi:  46nMAssay Description:Binding affinity by its ability to displace [3H]DPDPE from delta receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285003(3,10-dimethoxy-17-phenethyl-17-azatetracyclo[7.5.3...)
Affinity DataKi:  49nMAssay Description:Binding affinity by its ability to displace [3H]DPDPE from delta receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50148071((-)-N-(Cycloproylmethyl)-4,14-dimethoxymorphinan-6...)
Affinity DataKi:  61nMAssay Description:Binding affinity by its ability to displace [3H]-U-69,593 from kappa receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50148071((-)-N-(Cycloproylmethyl)-4,14-dimethoxymorphinan-6...)
Affinity DataKi:  105nMAssay Description:Binding affinity by its ability to displace [3H]DPDPE from delta receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50285003(3,10-dimethoxy-17-phenethyl-17-azatetracyclo[7.5.3...)
Affinity DataKi:  690nMAssay Description:Binding affinity by its ability to displace [3H]-U-69,593 from kappa receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article