Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50034863
LigandPNGBDBM50288462((R)-2-{(2R,5S)-2-[(R)-3-((R)-2-Carboxy-pyrrolidine...)
Affinity DataIC50:  0.25nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288477(3-(1-carbamoyl-2-phenylethylcarbamoyl)-3-[1-[7-oxo...)
Affinity DataIC50:  0.700nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288474((S)-1-(2-{(2-Cyclohexyl-ethyl)-[(S)-2-(2-1H-indol-...)
Affinity DataIC50:  0.940nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288473((S)-1-(2-{(2-Cyclohexyl-ethyl)-[(S)-2-(2-1H-indol-...)
Affinity DataIC50:  2.30nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288465((S)-1-(2-{(2-Cyclohexyl-ethyl)-[(S)-2-(2-1H-indol-...)
Affinity DataIC50:  17nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288463((R)-2-{(2R,5S)-2-[(R)-3-(Carboxymethyl-carbamoyl)-...)
Affinity DataIC50:  27nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288475((S)-1-(2-{Cyclohexylmethyl-[(S)-2-(2-1H-indol-3-yl...)
Affinity DataIC50:  30nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288466((S)-1-(2-{[(S)-2-(2-1H-Indol-3-yl-acetylamino)-hex...)
Affinity DataIC50:  34nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288470((R)-2-[(2R,5S)-2-((R)-3-Carboxymethyl-3,4-dihydro-...)
Affinity DataIC50:  35nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288462((R)-2-{(2R,5S)-2-[(R)-3-((R)-2-Carboxy-pyrrolidine...)
Affinity DataIC50:  36nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288468(CHEMBL101313 | CHEMBL3142755 | N-(1-Carbamoyl-2-ph...)
Affinity DataIC50:  38nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288471((R)-2-[(2R,5S)-1-((R)-1-tert-Butoxycarbonyl-2,3-di...)
Affinity DataIC50:  39nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288467((R)-2-[(2R,5S)-2-(3,4-Dihydro-1H-isoquinoline-2-ca...)
Affinity DataIC50:  52nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288464((S)-2-(2-1H-Indol-3-yl-acetylamino)-hexanoic acid ...)
Affinity DataIC50:  146nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288476(CHEMBL100762 | {[(S)-2-(2-1H-Indol-3-yl-acetylamin...)
Affinity DataIC50:  165nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288472((R)-2-[(2R,5S)-2-((R)-3-Carbamoyl-3,4-dihydro-1H-i...)
Affinity DataIC50:  170nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288466((S)-1-(2-{[(S)-2-(2-1H-Indol-3-yl-acetylamino)-hex...)
Affinity DataIC50:  300nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50288469(CHEMBL103713 | {(2-Cyclohexyl-ethyl)-[(S)-2-(2-1H-...)
Affinity DataIC50:  370nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288463((R)-2-{(2R,5S)-2-[(R)-3-(Carboxymethyl-carbamoyl)-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288474((S)-1-(2-{(2-Cyclohexyl-ethyl)-[(S)-2-(2-1H-indol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288462((R)-2-{(2R,5S)-2-[(R)-3-((R)-2-Carboxy-pyrrolidine...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288475((S)-1-(2-{Cyclohexylmethyl-[(S)-2-(2-1H-indol-3-yl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288462((R)-2-{(2R,5S)-2-[(R)-3-((R)-2-Carboxy-pyrrolidine...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288473((S)-1-(2-{(2-Cyclohexyl-ethyl)-[(S)-2-(2-1H-indol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288472((R)-2-[(2R,5S)-2-((R)-3-Carbamoyl-3,4-dihydro-1H-i...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288471((R)-2-[(2R,5S)-1-((R)-1-tert-Butoxycarbonyl-2,3-di...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288470((R)-2-[(2R,5S)-2-((R)-3-Carboxymethyl-3,4-dihydro-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288464((S)-2-(2-1H-Indol-3-yl-acetylamino)-hexanoic acid ...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288467((R)-2-[(2R,5S)-2-(3,4-Dihydro-1H-isoquinoline-2-ca...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288465((S)-1-(2-{(2-Cyclohexyl-ethyl)-[(S)-2-(2-1H-indol-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50288469(CHEMBL103713 | {(2-Cyclohexyl-ethyl)-[(S)-2-(2-1H-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for displacement of [3H]-L-364,718 from Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In DepthDetails Article