Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50034947
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450653(CHEMBL2115493)
Affinity DataIC50: 0.00500nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450653(CHEMBL2115493)
Affinity DataIC50: 0.0100nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450656(CHEMBL2114469)
Affinity DataIC50: 0.0100nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450656(CHEMBL2114469)
Affinity DataIC50: 0.0400nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071201((R)-2-[(R)-2-(2-{(R)-2-[(R)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 0.0710nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450653(CHEMBL2115493)
Affinity DataIC50: 0.25nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071201((R)-2-[(R)-2-(2-{(R)-2-[(R)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50007329(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 0.600nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM21130(U69,593 | N-methyl-N-(7-(1-pyrrolidinyl)-1-oxaspir...)
Affinity DataIC50: 0.630nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 0.630nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450655(CHEMBL2114470)
Affinity DataIC50: 1nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50007329(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 1.80nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450655(CHEMBL2114470)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450656(CHEMBL2114469)
Affinity DataIC50: 2.5nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataIC50: 3nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 4nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071201((R)-2-[(R)-2-(2-{(R)-2-[(R)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 6.30nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450654(CHEMBL2115492)
Affinity DataIC50: 10nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450654(CHEMBL2115492)
Affinity DataIC50: 10nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071199((R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 50nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450655(CHEMBL2114470)
Affinity DataIC50: 50nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071199((R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071199((R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 158nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450654(CHEMBL2115492)
Affinity DataIC50: 320nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50007329(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 400nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071202((R)-2-[(R)-2-(2-{(S)-2-[(R)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071202((R)-2-[(R)-2-(2-{(S)-2-[(R)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450653(CHEMBL2115493)
Affinity DataIC50: 6.31E+3nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450656(CHEMBL2114469)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450655(CHEMBL2114470)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071202((R)-2-[(R)-2-(2-{(S)-2-[(R)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against rat mu-opioid receptor expressed in CHO cells by competitive inhibition of 1 nM [3H]DAMGOMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071199((R)-2-[(R)-2-(2-{2-[(R)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071202((R)-2-[(R)-2-(2-{(S)-2-[(R)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50450654(CHEMBL2115492)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
Institute For Bioorganic Research

Curated by ChEMBL
LigandPNGBDBM50071201((R)-2-[(R)-2-(2-{(R)-2-[(R)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed