TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 340nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 580nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 870nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.02E+3nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 790nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 880nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 960nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 990nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute Of Bio-Science And Technology
Curated by ChEMBL
Institute Of Bio-Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair