Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50045518
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50008072((3S-cis)-3-ethyldihydro-4-[(1-methyl-1H-imidazol-5...)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50066079(Milameline)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50066076(CHEMBL3402921)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50066078(CHEMBL3402923)
Affinity DataEC50:  780nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50066074(CHEMBL3402918)
Affinity DataEC50:  5.68E+3nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50066075(CHEMBL3402919)
Affinity DataEC50:  7.54E+3nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50066077(CHEMBL3402922)
Affinity DataEC50:  1.73E+4nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataEC50:  1.00E+5nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2016
Entry Details Article
PubMed