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Found 12 Enz. Inhib. hit(s) with all data for entry = 50047812
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191108(CHEMBL3974458)
Affinity DataIC50:  0.920nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50112086(3-({2-[(4-Carbamimidoyl-phenylamino)-methyl]-1-met...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191077(CHEMBL3953757)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191112(CHEMBL3902879)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191076(CHEMBL3903935)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191074(CHEMBL3954784)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191197(CHEMBL3982468)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191109(CHEMBL3974821)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191075(CHEMBL3930866)
Affinity DataIC50:  5nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191110(CHEMBL3927138)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191073(CHEMBL3947048)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Shanghai Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50191111(CHEMBL3936103)
Affinity DataIC50:  16nMAssay Description:Inhibition of human thrombin pre-incubated for 10 mins before Ac-FVR-AMC substrate addition and measured after 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed