Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50048631
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  27nMAssay Description:Concentration required to inhibit [3H]naltrexone binding to Opioid receptorsMore data for this Ligand-Target Pair
LigandPNGBDBM50003560(4-methoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.0...)
Affinity DataIC50:  2.00E+3nMAssay Description:Concentration required to inhibit [3H]naltrexone binding to Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223879(CHEMBL280688)
Affinity DataIC50:  3.00E+3nMAssay Description:Concentration required to inhibit [3H]naltrexone binding to Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50017233(CHEMBL592 | LEVO-DROMORAN | LEVORPHANOL)
Affinity DataIC50:  4.00E+3nMAssay Description:Concentration required to inhibit [3H]naltrexone binding to Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50019351((-)-Codeine | (Codeine) | (codeine)10-methoxy-4-me...)
Affinity DataIC50:  1.00E+4nMAssay Description:Concentration required to inhibit [3H]naltrexone binding to Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223878(CHEMBL22919)
Affinity DataIC50:  2.00E+4nMAssay Description:Concentration required to inhibit [3H]naltrexone binding to Opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed