Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50049110
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234609BDBM50234609(Cariporide | HOE-642)
Affinity DataIC50: 172nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234607BDBM50234607(CHEMBL4071353)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234598BDBM50234598(CHEMBL4095965)
Affinity DataIC50: 5.09E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 32701BDBM32701(MLS000529214 | cid_570059 | SMR000121689 | Benzotr...)
Affinity DataIC50: 5.16E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234612BDBM50234612(CHEMBL4082866)
Affinity DataIC50: 5.92E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234601BDBM50234601(CHEMBL4072374)
Affinity DataIC50: 6.06E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234602BDBM50234602(CHEMBL557236)
Affinity DataIC50: 6.35E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234616BDBM50234616(CHEMBL4074684)
Affinity DataIC50: 6.51E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 16173BDBM16173(3,5-diamino-N-carbamimidoyl-6-chloropyrazine-2-car...)
Affinity DataIC50: 6.67E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234604BDBM50234604(CHEMBL425230)
Affinity DataIC50: 6.81E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234614BDBM50234614(CHEMBL4084954)
Affinity DataIC50: 6.98E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234610BDBM50234610(CHEMBL204234)
Affinity DataIC50: 7.24E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234596BDBM50234596(CHEMBL1884989)
Affinity DataIC50: 7.25E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234606BDBM50234606(CHEMBL4097403)
Affinity DataIC50: 8.65E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234617BDBM50234617(CHEMBL3086212)
Affinity DataIC50: 9.71E+4nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234603BDBM50234603(CHEMBL4072288)
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234615BDBM50234615(CHEMBL4063302)
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234605BDBM50234605(CHEMBL4087253)
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234600BDBM50234600(CHEMBL4093129)
Affinity DataIC50: 1.55E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234599BDBM50234599(CHEMBL4100842)
Affinity DataIC50: 1.57E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234608BDBM50234608(CHEMBL4068558)
Affinity DataIC50: 1.77E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234611BDBM50234611(CHEMBL4085368)
Affinity DataIC50: 1.91E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234613BDBM50234613(CHEBI:75331 | 1H-Benzo[D][1,2,3]Triazole | 1H-Benz...)
Affinity DataIC50: 1.93E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed
TargetSodium/hydrogen exchanger 1(Human)
Punjabi University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50234597BDBM50234597(CHEMBL4079373)
Affinity DataIC50: 3.55E+5nMAssay Description:Inhibition of platelet NHE1 in human platelet rich plasma assessed as decrease in platelet swelling preincubated for 3 mins followed by sodium propio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details Article
PubMed