Compile Data Set for Download or QSAR
maximum 50k data
Found 112 Enz. Inhib. hit(s) with all data for entry = 7408
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193349(US9199927, 108 | US9199927, 60)
Affinity DataIC50:  0.140nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193350(US9199927, 61)
Affinity DataIC50:  0.140nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193351(US9199927, 62)
Affinity DataIC50:  0.170nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193290(US9199927, 1)
Affinity DataIC50:  0.170nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193310(US9199927, 21)
Affinity DataIC50:  0.170nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193313(US9199927, 24)
Affinity DataIC50:  0.170nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193317(US9199927, 28)
Affinity DataIC50:  0.170nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193360(US9199927, 71)
Affinity DataIC50:  0.180nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193315(US9199927, 26)
Affinity DataIC50:  0.180nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193349(US9199927, 108 | US9199927, 60)
Affinity DataIC50:  0.190nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193290(US9199927, 1)
Affinity DataIC50:  0.190nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193304(US9199927, 15)
Affinity DataIC50:  0.190nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193316(US9199927, 27)
Affinity DataIC50:  0.190nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193319(US9199927, 30)
Affinity DataIC50:  0.190nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193304(US9199927, 15)
Affinity DataIC50:  0.200nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193311(US9199927, 22)
Affinity DataIC50:  0.200nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193318(US9199927, 29)
Affinity DataIC50:  0.210nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193349(US9199927, 108 | US9199927, 60)
Affinity DataIC50:  0.210nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193369(US9199927, 80)
Affinity DataIC50:  0.210nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193349(US9199927, 108 | US9199927, 60)
Affinity DataIC50:  0.210nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193313(US9199927, 24)
Affinity DataIC50:  0.210nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193414(US9199927, 96)
Affinity DataIC50:  0.220nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193303(US9199927, 14)
Affinity DataIC50:  0.220nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193350(US9199927, 61)
Affinity DataIC50:  0.230nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193303(US9199927, 14)
Affinity DataIC50:  0.230nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193360(US9199927, 71)
Affinity DataIC50:  0.230nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193305(US9199927, 16)
Affinity DataIC50:  0.230nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193395(US9199927, 113)
Affinity DataIC50:  0.240nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193323(US9199927, 34)
Affinity DataIC50:  0.240nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193317(US9199927, 28)
Affinity DataIC50:  0.240nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193314(US9199927, 25)
Affinity DataIC50:  0.25nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193310(US9199927, 21)
Affinity DataIC50:  0.260nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193316(US9199927, 27)
Affinity DataIC50:  0.260nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193319(US9199927, 30)
Affinity DataIC50:  0.260nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193305(US9199927, 16)
Affinity DataIC50:  0.260nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193306(US9199927, 17)
Affinity DataIC50:  0.270nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193348(US9199927, 59)
Affinity DataIC50:  0.270nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193324(US9199927, 35)
Affinity DataIC50:  0.280nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193312(US9199927, 23)
Affinity DataIC50:  0.280nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193395(US9199927, 113)
Affinity DataIC50:  0.280nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193311(US9199927, 22)
Affinity DataIC50:  0.290nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193314(US9199927, 25)
Affinity DataIC50:  0.290nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193415(US9199927, 102)
Affinity DataIC50:  0.290nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193351(US9199927, 62)
Affinity DataIC50:  0.290nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193315(US9199927, 26)
Affinity DataIC50:  0.290nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193369(US9199927, 80)
Affinity DataIC50:  0.300nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193341(US9199927, 52)
Affinity DataIC50:  0.300nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193415(US9199927, 102)
Affinity DataIC50:  0.300nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTrypsinogen 16(Mus musculus (Mouse))
Astellas Pharma

US Patent
LigandPNGBDBM193330(US9199927, 41)
Affinity DataIC50:  0.310nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine protease 1(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM193320(US9199927, 31)
Affinity DataIC50:  0.310nMpH: 8.0 T: 2°CAssay Description:The compound was dissolved in dimethyl sulfoxide (DMSO), and diluted to an arbitrary concentration (A). A was 100-fold diluted with a buffer (0.1 M T...More data for this Ligand-Target Pair
In DepthDetails US Patent
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