Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 1493
TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326336BDBM326336(US9662310, Example 1 | US9662310, Example 28 | (1R...)
Affinity DataIC50: 4.5nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326397BDBM326397((1R,2S)-2-[(2R)-2-(Aminomethyl)butyl]-1-(1-phenyl-...)
Affinity DataIC50: 7.90nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326395BDBM326395((1R,2S)-2-[(2R)-2-(Aminomethyl)butyl]-1-(1-pyridin...)
Affinity DataIC50: 8.30nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326393BDBM326393((1R,2S)-2-[(2R)-3-Amino-2-methylpropyl]-1-[1-(5-me...)
Affinity DataIC50: 8.70nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326336BDBM326336(US9662310, Example 1 | US9662310, Example 28 | (1R...)
Affinity DataIC50: 8.70nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326383BDBM326383((1R,2S)-2-(3-Aminopropyl)-1-(1-pyridin-2-yl-1H-imi...)
Affinity DataIC50: 11nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326389BDBM326389((1R,2S)-2-[(2R)-3-Amino-2-methylpropyl]-1-(1-pyrid...)
Affinity DataIC50: 11nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326398BDBM326398((1R,2S)-2-[ | US9662310, Example 63)
Affinity DataIC50: 12nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326403BDBM326403(2-[(2R)-4-Aminobutane-2-yl]-1-[1-(pyridin-2-yl)-1H...)
Affinity DataIC50: 12nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326365BDBM326365(US9662310, Example 30 | US9662310, Example 31 | (1...)
Affinity DataIC50: 13nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326388BDBM326388((1R,2S)-2-[(2-Aminomethyl)butyl]-1-(1-phenyl-1H-im...)
Affinity DataIC50: 13nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326385BDBM326385((1R,2S)-2-[(2R)-3-Amino-2-methylpropyl]-1-(1-pheny...)
Affinity DataIC50: 14nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326340BDBM326340((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(trans-4-methylcy...)
Affinity DataIC50: 14nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326365BDBM326365(US9662310, Example 30 | US9662310, Example 31 | (1...)
Affinity DataIC50: 15nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326379BDBM326379((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(5-methoxypyridin...)
Affinity DataIC50: 16nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326381BDBM326381((1R*,2S*)-2-(3-Aminopropyl)-1-(1-isoquinolin-3-yl-...)
Affinity DataIC50: 16nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326342BDBM326342((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(4-methylphenyl)-...)
Affinity DataIC50: 16nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326384BDBM326384((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(5-methylpyridin-...)
Affinity DataIC50: 18nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326376BDBM326376((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(5-fluoropyridin-...)
Affinity DataIC50: 19nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326399BDBM326399((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(4-methylpyridin-...)
Affinity DataIC50: 19nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326350BDBM326350((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(4-fluorophenyl)-...)
Affinity DataIC50: 21nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326353BDBM326353((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(4-chlorophenyl)-...)
Affinity DataIC50: 25nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326378BDBM326378((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(1-benzofuran-5-y...)
Affinity DataIC50: 26nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326341BDBM326341((1R*,2S*)-2-(3-Aminopropyl)-1-(1-phenyl-1H-imidazo...)
Affinity DataIC50: 27nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326356BDBM326356((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(2-naphthyl)-1H-i...)
Affinity DataIC50: 27nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326360BDBM326360((1R*,2S*)-2-(3-Aminopropyl)-1-(1-pyridin-2-yl-1H-i...)
Affinity DataIC50: 29nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326339BDBM326339((1R*,2S*)-2-(3-Aminopropyl)-1-(1-cyclohexyl-1H-imi...)
Affinity DataIC50: 29nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326375BDBM326375((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(4-cyanophenyl)-1...)
Affinity DataIC50: 29nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326374BDBM326374((1R*,2S*)-2-(3-Aminopropyl)-1-(1-pyrimidin-2-yl-1H...)
Affinity DataIC50: 30nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326346BDBM326346((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(4-ethylphenyl)-1...)
Affinity DataIC50: 31nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326391BDBM326391((1R,2S)-2-[(2S)-3-Amino-2-methylpropyl]-1-(1-pyrid...)
Affinity DataIC50: 33nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326367BDBM326367((1R*,2S*)-2-(3-Amino-2-methylpropyl)-1-(1-phenyl-1...)
Affinity DataIC50: 35nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326386BDBM326386((1R,2S)-2-[(2S)-3-Amino-2-methylpropyl]-1-(1-pheny...)
Affinity DataIC50: 35nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326347BDBM326347((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(4-methoxyphenyl)...)
Affinity DataIC50: 36nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326371BDBM326371((1R*,2R*)-2-(3-Amino-1-methylpropyl)-1-(1-phenyl-1...)
Affinity DataIC50: 36nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326343BDBM326343((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(3-methylphenyl)-...)
Affinity DataIC50: 37nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326368BDBM326368((1R*,2S*)-2-(3-Amino-2-methylpropyl)-1-[1-(4-methy...)
Affinity DataIC50: 39nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326357BDBM326357((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(3-fluorophenyl)-...)
Affinity DataIC50: 40nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326401BDBM326401((1R,2S)-2-[(2R)-2-(Aminomethyl)pentyl]-1-(1-pyridi...)
Affinity DataIC50: 41nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326345BDBM326345((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(3,4-dimethylphen...)
Affinity DataIC50: 42nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326351BDBM326351((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(4-phenoxyphenyl)...)
Affinity DataIC50: 52nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326382BDBM326382((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(1-naphthyl)-1H-i...)
Affinity DataIC50: 54nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326377BDBM326377((1R*,2S*)-2-(3-Aminopropyl)-1-(1-quinolin-2-yl-1H-...)
Affinity DataIC50: 58nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326373BDBM326373((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(1,3-thiazol-2-yl...)
Affinity DataIC50: 58nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326352BDBM326352((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(3,4-difluorophen...)
Affinity DataIC50: 61nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326380BDBM326380((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(5-chloropyridin-...)
Affinity DataIC50: 63nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326354BDBM326354((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(3-chlorophenyl)-...)
Affinity DataIC50: 70nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326400BDBM326400((1R*,2S*)-2-(3-Aminopropyl)-1-[1-(6-methylpyridin-...)
Affinity DataIC50: 73nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326338BDBM326338((1R*,2S*)-2-(3-Aminopropyl)-1-(1-propyl-1H-imidazo...)
Affinity DataIC50: 97nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

TargetCarboxypeptidase B2(Human)
Daiichi Sankyo

US Patent
LigandChemical structure of BindingDB Monomer ID 326359BDBM326359((1R*,2S*)-2-(3-Aminopropyl)-1-(1-pyridin-3-yl-1H-i...)
Affinity DataIC50: 98nMAssay Description:HEPES buffered saline (20 mM HEPES, 150 mM NaCl, pH 7.4; hereinafter, referred to as HBS) was used in the preparation of a reaction solution. To 12 &...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details
US Patent

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