Compile Data Set for Download or QSAR
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Found 18 Enz. Inhib. hit(s) with all data for entry = 50036347
TargetMu-type opioid receptor(GUINEA PIG)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032527(17-cyclopropylmethyl-10-ethoxy-4-hydroxy-3-methoxy...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity was evaluated by measuring the ability to displace [3H]DAMGO radioligand binding from Opioid receptor mu 1 in guinea pig brain membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032530(17-cyclopropylmethyl-4-hydroxy-3,10-dimethoxy-17-a...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity was evaluated by measuring the ability to displace [3H]U-69593 radioligand binding from Opioid receptor kappa 1 in guinea pig brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032527(17-cyclopropylmethyl-10-ethoxy-4-hydroxy-3-methoxy...)
Affinity DataKi:  5.5nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]U-69593 radioligand binding from Opioid receptor kappa 1 in guinea pi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032530(17-cyclopropylmethyl-4-hydroxy-3,10-dimethoxy-17-a...)
Affinity DataKi:  6.20nMAssay Description:Binding affinity was evaluated by measuring the ability to displace [3H]DAMGO radioligand binding from Opioid receptor mu 1 in guinea pig brain membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032526(17-allyl-4-hydroxy-3,10-dimethoxy-17-azatetracyclo...)
Affinity DataKi:  7.30nMAssay Description:Binding affinity was evaluated by measuring the ability to displace [3H]DAMGO radioligand binding from Opioid receptor mu 1 in guinea pig brain membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032528(3-butoxy-17-cyclopropylmethyl-4-hydroxy-10-methoxy...)
Affinity DataKi:  11nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]DAMGO radioligand binding from Opioid receptor mu 1 in guinea pig bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032528(3-butoxy-17-cyclopropylmethyl-4-hydroxy-10-methoxy...)
Affinity DataKi:  13nMAssay Description:Binding affinity was evaluated by measuring the ability to displace [3H]U-69593 radioligand binding from Opioid receptor kappa 1 in guinea pig brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032530(17-cyclopropylmethyl-4-hydroxy-3,10-dimethoxy-17-a...)
Affinity DataKi:  14nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]DPDPE radioligand binding from delta opioid receptor in guinea pig br...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032527(17-cyclopropylmethyl-10-ethoxy-4-hydroxy-3-methoxy...)
Affinity DataKi:  21nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]DPDPE radioligand binding from delta opioid receptor in guinea pig br...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032525(17-cyclopropylmethyl-4,10-dihydroxy-3-methoxy-17-a...)
Affinity DataKi:  23nMAssay Description:Binding affinity was evaluated by measuring the ability to displace [3H]U-69593 radioligand binding from Opioid receptor kappa 1 in guinea pig brain ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50148071((-)-N-(Cycloproylmethyl)-4,14-dimethoxymorphinan-6...)
Affinity DataKi:  24nMAssay Description:Binding affinity was evaluated by measuring the ability to displace [3H]DAMGO radioligand binding from Opioid receptor mu 1 in guinea pig brain membr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032526(17-allyl-4-hydroxy-3,10-dimethoxy-17-azatetracyclo...)
Affinity DataKi:  25nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]U-69593 radioligand binding from Opioid receptor kappa 1 in guinea pi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032526(17-allyl-4-hydroxy-3,10-dimethoxy-17-azatetracyclo...)
Affinity DataKi:  26nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]DPDPE radioligand binding from delta opioid receptor in guinea pig br...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032528(3-butoxy-17-cyclopropylmethyl-4-hydroxy-10-methoxy...)
Affinity DataKi:  42nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]DPDPE radioligand binding from delta opioid receptor in guinea pig br...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032525(17-cyclopropylmethyl-4,10-dihydroxy-3-methoxy-17-a...)
Affinity DataKi:  54nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]DAMGO radioligand binding from Opioid receptor mu 1 in guinea pig bra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50148071((-)-N-(Cycloproylmethyl)-4,14-dimethoxymorphinan-6...)
Affinity DataKi:  61nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]DPDPE radioligand binding from delta opioid receptor in guinea pig br...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50148071((-)-N-(Cycloproylmethyl)-4,14-dimethoxymorphinan-6...)
Affinity DataKi:  105nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]U-69593 radioligand binding from Opioid receptor kappa 1 in guinea pi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50032525(17-cyclopropylmethyl-4,10-dihydroxy-3-methoxy-17-a...)
Affinity DataKi:  334nMAssay Description:In vivo binding affinity was evaluated by measuring the ability to displace [3H]DPDPE radioligand binding from delta opioid receptor in guinea pig br...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed