Compile Data Set for Download or QSAR
maximum 50k data
Found 48 Enz. Inhib. hit(s) with all data for entry = 50005160
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  0.300nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  0.5nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033640(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  2nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033640(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  2nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033640(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  7nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  8nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033629(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  10nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  12nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033629(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  14nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  23nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033629(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  32nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  42nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  57nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  65nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (% of amylase secretion at 1 mM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  75nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  190nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  200nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  205nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  210nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  250nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033631(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  500nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1.75E+3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033636(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033629(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  20nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50016425((S)-3-{(S)-2-[(S)-2-(2-{(S)-2-[(S)-2-tert-Butoxyca...)
Affinity DataEC50:  0.0500nMAssay Description:Tested in vitro for amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  20nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033640(2-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  3nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033634(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  4nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  6nMAssay Description:Tested for inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033632(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  22nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Homo sapiens (Human))
Ep Cnrs 51

Curated by ChEMBL
LigandPNGBDBM50033633(3-{2-[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-sul...)
Affinity DataEC50:  50nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (percent of secretion)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed