Compile Data Set for Download or QSAR
Report error Found 1363 Enz. Inhib. hit(s) with all data for entry = 2051
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353376BDBM353376(4-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]p...)
Affinity DataIC50: 4nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167699BDBM167699(US9073922, 186 | US9796708, Example 186)
Affinity DataIC50: 4nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353374BDBM353374(N-methyl-4-[2-(1,2,3,6-tetrahydropyridin-4-yl)-1H-...)
Affinity DataIC50: 6nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353253BDBM353253(4-(5-fluoro-2-methoxyphenyl)-2-(1,2,5,6-tetrahydro...)
Affinity DataIC50: 7nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167716BDBM167716(US9073922, 203 | US9796708, Example 203)
Affinity DataIC50: 8nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167703BDBM167703(US9073922, 190 | US9796708, Example 190)
Affinity DataIC50: 8nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353138BDBM353138(4-fluoro-N-(4-fluorobenzyl)-3-[2-(piperidin-4-yl)-...)
Affinity DataIC50: 9nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353195BDBM353195(3-[4-(4-{2-fluoro-5-[(3-fluorobenzyl)amino]phenyl}...)
Affinity DataIC50: 9nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167553BDBM167553(US9073922, 37 | US9796708, Example 37)
Affinity DataIC50: 10nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167602BDBM167602(US9073922, 87 | US9796708, Example 87)
Affinity DataIC50: 10nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353433BDBM353433(3-chloro-4-(5-fluoro-2-methoxyphenyl)-2-(1,2,3,6-t...)
Affinity DataIC50: 10nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167533BDBM167533(US9073922, 17 | US9796708, Example 17)
Affinity DataIC50: 11nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167719BDBM167719(US9073922, 206 | US9796708, Example 206)
Affinity DataIC50: 11nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167659BDBM167659(US9073922, 146 | US9796708, Example 146)
Affinity DataIC50: 12nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167538BDBM167538(US9073922, 22 | US9796708, Example 22)
Affinity DataIC50: 12nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167616BDBM167616(US9073922, 102 | US9796708, Example 102)
Affinity DataIC50: 12nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353375BDBM353375(5-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]p...)
Affinity DataIC50: 12nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167619BDBM167619(US9073922, 105 | US9796708, Example 105)
Affinity DataIC50: 13nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167611BDBM167611(US9073922, 97 | US9796708, Example 97)
Affinity DataIC50: 14nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167642BDBM167642(US9073922, 129 | US9796708, Example 129)
Affinity DataIC50: 14nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167626BDBM167626(US9073922, 112 | US9796708, Example 112)
Affinity DataIC50: 14nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353767BDBM353767(US9796708, Example 999 | 2-{4-[4-(5-fluoro-2-metho...)
Affinity DataIC50: 14nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353124BDBM353124(4-fluoro-N-[4-(methylsulfonyl)benzyl]-3-[2-(piperi...)
Affinity DataIC50: 14nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167567BDBM167567(US9073922, 52 | US9796708, Example 52)
Affinity DataIC50: 14nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353113BDBM353113(N-benzyl-2,4-difluoro-5-[2-(piperidin-4-yl)-1H-pyr...)
Affinity DataIC50: 14nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167549BDBM167549(US9073922, 33 | US9796708, Example 33)
Affinity DataIC50: 15nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353139BDBM353139(4-[({4-fluoro-3-[2-(piperidin-4-yl)-1H-pyrrolo[2,3...)
Affinity DataIC50: 15nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353142BDBM353142(4-fluoro-N-[3-(methylsulfonyl)benzyl]-3-[2-(piperi...)
Affinity DataIC50: 15nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167520BDBM167520(US9073922, 4 | US9796708, Example 4)
Affinity DataIC50: 15nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167572BDBM167572(US9073922, 57 | US9796708, Example 57)
Affinity DataIC50: 15nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167571BDBM167571(US9073922, 56 | US9796708, Example 56)
Affinity DataIC50: 15nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167577BDBM167577(US9073922, 62 | US9796708, Example 62)
Affinity DataIC50: 15nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167669BDBM167669(US9073922, 156 | US9796708, Example 156)
Affinity DataIC50: 15nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353426BDBM353426(4-(4-fluoro-2-methoxyphenyl)-2-(1,2,3,6-tetrahydro...)
Affinity DataIC50: 16nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167517BDBM167517(US9073922, 1 | US9796708, Example 1)
Affinity DataIC50: 16nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353377BDBM353377(4-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]p...)
Affinity DataIC50: 16nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353095BDBM353095(2-(2,5-dihydro-1H-pyrrol-3-yl)-4-(5-fluoro-2-metho...)
Affinity DataIC50: 16nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167723BDBM167723(US9073922, 210 | US9796708, Example 210)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167663BDBM167663(US9073922, 150 | US9796708, Example 150)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353140BDBM353140(3-[({4-fluoro-3-[2-(piperidin-4-yl)-1H-pyrrolo[2,3...)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353252BDBM353252(N-(3,5-difluorobenzyl)-4-fluoro-3-[2-(1,2,3,6-tetr...)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167552BDBM167552(US9073922, 36 | US9796708, Example 36)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353438BDBM353438(4-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]p...)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353439BDBM353439(4-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]p...)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353212BDBM353212(5-fluoro-4-(5-fluoro-2-methoxyphenyl)-2-(piperidin...)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167574BDBM167574(US9073922, 59 | US9796708, Example 59)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 353389BDBM353389(3-bromo-4-(5-fluoro-2-methoxyphenyl)-2-(1,2,3,6-te...)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167544BDBM167544(US9073922, 28 | US9796708, Example 28)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167591BDBM167591(US9073922, 76 | US9796708, Example 76)
Affinity DataIC50: 17nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Abbvie

US Patent
LigandChemical structure of BindingDB Monomer ID 167724BDBM167724(US9073922, 211 | US9796708, Example 211)
Affinity DataIC50: 18nMAssay Description:CDK9 enzyme activities were measured using LANCE ULight TR-FRET kinase assay reagents (PerkinElmer, Waltham, Mass.). Compounds were directly added in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2019
Entry Details
US Patent

Displayed 1 to 50 (of 1363 total ) | Next | Last >>
Jump to: