Compile Data Set for Download or QSAR
maximum 50k data
Found 125 Enz. Inhib. hit(s) with all data for entry = 2063
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329827((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(trimet...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329828((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(3-(pyrid...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329829((rac)-[(1R,2R,3S,4R)-4-{[2-(9H-carbazol-3-yl)pyraz...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329830((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(5-methyl...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329831((rac)-((1R,2R,3S,4R)-4-(2-(7-chloroquinolin-4-yl)p...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329832((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(3-(trifl...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329833((rac)-((1R,2R,3S,4R)-4-(2-(3,3-dimethyl-2,3-dihydr...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329834((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(quinolin-...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329835((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(quinolin-...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329836((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(triflu...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329837((rac)-((1R,2R,3S,4R)-4-((2-(Benzo[b]thiophen-7-yl)...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329838((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(pyrrol...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329839((rac)-(1R,2R,3S,4R)-4-(2-(3-cyclopentenylphenyl)py...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329840((rac)-[(1R,2R,3S,4R)-4-{[2-(3-cyclopentylphenyl)py...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329841((rac)-((1R,2R,3S,4R)-4-(2-(benzofuran-3-yl)pyrazol...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329842((rac)-((1R,2R,3S,4R)-4-((2-(3-(Difluoromethoxy)phe...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329844((rac)-((1R,2R,3S,4R)-4-(2-(6-tert-butylpyridin-2-y...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329845((rac)-((1R,2R,3S,4R)-4-(2-(3,3-dimethyl-1,3-dihydr...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329846((rac)-[(1R,2R,3S,4R)-4-{[2-(5-chloro-1H-indol-3-yl...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329847((rac)-[(1R,2R,3S,4R)-4-{[2-(6-chloro-1H-indol-3-yl...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329848((rac)-((1R,2R,3S,4R)-4-((2-(Dibenzo[b,d]thiophen-4...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329849((rac)-((1R,2R,3S,4R)-4-(2-(5-chloro-2-(trifluorome...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329850((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(1,1,1-...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329853((rac)-((1R,2R,3S,4R)-4-((2-(Benzo[b]thiophen-4-yl)...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329854((rac)-[(1R,2R,3S,4R)-4-{[2-(9H-carbazol-2-yl)pyraz...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM347108(US10202389, Compound I-063 | US10202389, Example 9...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329857((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329858((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329910((s.e.)-((1R,2R,3S,4R)-4-(2-(4-fluoronaphthalen-2-y...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329911((s.e.)-((1R,2R,3S,4R)-4-(2-(1-fluoronaphthalen-2-y...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329912((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methox...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329913((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(6-phenyl...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329914((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-({2-[3-(1-met...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329915((rac)-{(1R,2R,3S,4R)-4-[(2-{3-[2-chloro-1-(hydroxy...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329794((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(1-naphth...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329795((rac)((1R,2R,3S,4R)-4-(2-(biphenyl-3-yl)pyrazolo[1...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329797((rac)-((1R,2R,3S,4R)-4-((2-(3-Chlorophenyl)pyrazol...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329799((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(3-(trifl...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329802((rac)-((1R,2R,3S,4R)-4-(2-(dibenzo[b,d]furan-4-yl)...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329807((rac)-((1R,2R,3S,4R)-4-((2-(3-(tert-Butyl)phenyl)p...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329859((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(2-phenyl...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329862((rac)-((1R,2R,3S,4R)-4-(2-(4-fluoro-2-methoxypheny...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329863((rac)-((1R,2R,3S,4R)-4-(2-(5-chlorobenzo[b]thiophe...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329864((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methoyp...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329867((rac)-((1R,2R,3S,4R)-4-(2-(1H-indol-4-yl)pyrazolo[...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329868((rac)-((1R,2R,3S,4R)-4-(2-(3-(cyclopropylmethylthi...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329869((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(piperi...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329870((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-morphol...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329873((rac)-((1R,2R,3S,4R)-4-(2-(5-fluorobenzo[b]thiophe...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSUMO-activating enzyme subunit 2(Homo sapiens (Human))
Millennium Pharmaceuticals

US Patent
LigandPNGBDBM329874((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-meth...)
Affinity DataIC50: <10nMAssay Description:he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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