Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50007599
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065173((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 8nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065188((S)-N-(2-Cyclohexyl-ethyl)-3-{2-[ethyl-(4-piperidi...)
Affinity DataIC50: 10nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065174((S)-N-((R)-1-Carboxy-3-cyclohexyl-propyl)-3-{2-[et...)
Affinity DataIC50: 11nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065185((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 11nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065177((S)-N-[(S)-1-Carboxy-2-(decahydro-naphthalen-1-yl)...)
Affinity DataIC50: 11nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065167((S)-N-((R)-2-Cyclohexyl-1-ethoxycarbonyl-ethyl)-3-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: 17nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065177((S)-N-[(S)-1-Carboxy-2-(decahydro-naphthalen-1-yl)...)
Affinity DataIC50: 19nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065172((S)-N-((S)-1-Carboxy-2-naphthalen-2-yl-ethyl)-3-{2...)
Affinity DataIC50: 22nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065182((S)-N-((S)-1-Carboxy-2-naphthalen-1-yl-ethyl)-3-{2...)
Affinity DataIC50: 22nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: 26nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065173((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 27nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065166((S)-N-((R)-1-Carbamoyl-2-cyclohexyl-ethyl)-3-{2-[e...)
Affinity DataIC50: 28nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065174((S)-N-((R)-1-Carboxy-3-cyclohexyl-propyl)-3-{2-[et...)
Affinity DataIC50: 31nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065180((S)-N-((R)-Carboxy-cyclohexyl-methyl)-3-{2-[ethyl-...)
Affinity DataIC50: 32nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065186((S)-N-((R)-1-Carboxy-2-cycloheptyl-ethyl)-3-{2-[et...)
Affinity DataIC50: 32nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065181((S)-N-((R)-1-Carboxy-2-cyclopentyl-ethyl)-3-{2-[et...)
Affinity DataIC50: 47nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065184((R)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 53nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065178((S)-N-((S)-1-Carboxy-2-phenyl-ethyl)-3-{2-[ethyl-(...)
Affinity DataIC50: 64nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065167((S)-N-((R)-2-Cyclohexyl-1-ethoxycarbonyl-ethyl)-3-...)
Affinity DataIC50: 64nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065172((S)-N-((S)-1-Carboxy-2-naphthalen-2-yl-ethyl)-3-{2...)
Affinity DataIC50: 68nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065188((S)-N-(2-Cyclohexyl-ethyl)-3-{2-[ethyl-(4-piperidi...)
Affinity DataIC50: 72nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065168((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 72nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065176((S)-N-((R)-1-Carboxy-2-cyclooctyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: 78nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065168((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 82nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065183((S)-N-[(S)-1-Carboxy-2-(decahydro-naphthalen-2-yl)...)
Affinity DataIC50: 96nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065166((S)-N-((R)-1-Carbamoyl-2-cyclohexyl-ethyl)-3-{2-[e...)
Affinity DataIC50: 97nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065182((S)-N-((S)-1-Carboxy-2-naphthalen-1-yl-ethyl)-3-{2...)
Affinity DataIC50: 110nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065190((S)-N-((R)-2-Cyclohexyl-1-hydroxymethyl-ethyl)-3-{...)
Affinity DataIC50: 129nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065185((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 130nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065192((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(5-piperidin-4-yl...)
Affinity DataIC50: 210nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065169((R)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 260nMAssay Description:Inhibition of radiolabeled fibrinogen binding to activated human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065165((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(6-guanidino-hexa...)
Affinity DataIC50: 470nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065187((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(5-guanidino-pent...)
Affinity DataIC50: 630nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065169((R)-2-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl...)
Affinity DataIC50: 720nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065189((S)-2-((S)-3-Carboxy-2-{2-[ethyl-(3-piperidin-4-yl...)
Affinity DataIC50: 770nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065170((S)-2-{(S)-3-Carboxy-2-[2-(4-piperidin-4-yl-butyry...)
Affinity DataIC50: 1.06E+3nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065191((S)-N-((R)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: 1.37E+3nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065179((S)-2-{(S)-3-Carboxy-2-[2-(5-guanidino-pentanoylam...)
Affinity DataIC50: 2.30E+3nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065175(1-((S)-3-Carboxy-2-{2-[ethyl-(4-piperidin-4-yl-but...)
Affinity DataIC50: 3.41E+3nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241180(3-[2-(2-Amino-5-guanidino-pentanoylamino)-acetylam...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241181(Arg-Gly-Asp-Val | (2S)-2-[(2S)-2-{2-[(2S)-2-amino-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241180(3-[2-(2-Amino-5-guanidino-pentanoylamino)-acetylam...)
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241180(3-[2-(2-Amino-5-guanidino-pentanoylamino)-acetylam...)
Affinity DataIC50: 8.20E+4nMAssay Description:Ability to inhibit the aggregation of fixed human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50241180(3-[2-(2-Amino-5-guanidino-pentanoylamino)-acetylam...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: 1.01E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: 1.65E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065171((S)-N-((S)-1-Carboxy-2-cyclohexyl-ethyl)-3-{2-[eth...)
Affinity DataIC50: 1.75E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065174((S)-N-((R)-1-Carboxy-3-cyclohexyl-propyl)-3-{2-[et...)
Affinity DataIC50: 1.93E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065166((S)-N-((R)-1-Carbamoyl-2-cyclohexyl-ethyl)-3-{2-[e...)
Affinity DataIC50: 2.35E+6nMAssay Description:Inhibition of HUVEC adhesion to fibrinogen-coated platesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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