Affinity DataKi: 3.80nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]spiperone (Dopamine receptor D2) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]7-OH-DPAT binding to Dopamine receptor D3 in rat tissue homogen...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]7-OH-DPAT binding to Dopamine receptor D3 in rat tissue homogen...More data for this Ligand-Target Pair
Affinity DataKi: 16.4nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]SCH-23390 (Dopamine receptor D1) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]SCH-23390 (Dopamine receptor D1) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]SCH-23390 (Dopamine receptor D1) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 49.6nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]spiperone (Dopamine receptor D2) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]7-OH-DPAT binding to Dopamine receptor D3 in rat tissue homogen...More data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]spiperone (Dopamine receptor D2) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]spiperone (Dopamine receptor D2) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]SCH-23390 (Dopamine receptor D1) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]SCH-23390 (Dopamine receptor D1) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]spiperone (Dopamine receptor D2) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]spiperone (Dopamine receptor D2) binding to rat tissue homogena...More data for this Ligand-Target Pair
Affinity DataKi: 353nMAssay Description:Binding affinity which represents concentration giving half-maximal inhibition of [3H]SCH-23390 (Dopamine receptor D1) binding to rat tissue homogena...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Universita' Di Siena
Curated by ChEMBL
Universita' Di Siena
Curated by ChEMBL
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of dopamine uptake from dopamine uptake siteMore data for this Ligand-Target Pair