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Found 14 Enz. Inhib. hit(s) with all data for entry = 50007831
TargetNeutrophil elastase(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068280(5-Benzyloxycarbonylamino-pentanoic acid 1,1,3-trio...)
Affinity DataIC50:  1.44E+3nMAssay Description:Inhibitory activity was measured against human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068284(3-Benzyloxycarbonylamino-propionic acid 1,1,3-trio...)
Affinity DataIC50:  2.26E+3nMAssay Description:Inhibitory activity was measured against human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068298(4-Benzyloxycarbonylamino-benzoic acid 1,1,3-trioxo...)
Affinity DataIC50:  2.66E+3nMAssay Description:Inhibitory activity was measured against human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068280(5-Benzyloxycarbonylamino-pentanoic acid 1,1,3-trio...)
Affinity DataIC50: >1.20E+4nMAssay Description:Inhibitory activity was measured against trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068284(3-Benzyloxycarbonylamino-propionic acid 1,1,3-trio...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibitory activity was measured against thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068284(3-Benzyloxycarbonylamino-propionic acid 1,1,3-trio...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibitory activity was measured against urokinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068280(5-Benzyloxycarbonylamino-pentanoic acid 1,1,3-trio...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibitory activity was measured against thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068284(3-Benzyloxycarbonylamino-propionic acid 1,1,3-trio...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibitory activity was measured against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068298(4-Benzyloxycarbonylamino-benzoic acid 1,1,3-trioxo...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibitory activity was measured against thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068280(5-Benzyloxycarbonylamino-pentanoic acid 1,1,3-trio...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibitory activity was measured against urokinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068284(3-Benzyloxycarbonylamino-propionic acid 1,1,3-trio...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibitory activity was measured against plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068280(5-Benzyloxycarbonylamino-pentanoic acid 1,1,3-trio...)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibitory activity was measured against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1/Trypsin-2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068284(3-Benzyloxycarbonylamino-propionic acid 1,1,3-trio...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibitory activity was measured against trypsin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50068280(5-Benzyloxycarbonylamino-pentanoic acid 1,1,3-trio...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibitory activity was measured against plasmin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed