Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50034980
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069471BDBM50069471(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 7nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069458BDBM50069458(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 10nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069459BDBM50069459(Thiophene-3-carboxylic acid (7-bromo-2,3-dioxo-1,2...)
Affinity DataIC50: 10nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069483BDBM50069483(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 10nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069495BDBM50069495(N-(7-Chloro-2,3-dioxo-1,2,3,4-tetrahydro-quinoxali...)
Affinity DataIC50: 10nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069465BDBM50069465(Thiophene-2-carboxylic acid (7-bromo-2,3-dioxo-1,2...)
Affinity DataIC50: 10nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069482BDBM50069482(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 10nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069478BDBM50069478(3-Methyl-thiophene-2-carboxylic acid (7-bromo-2,3-...)
Affinity DataIC50: 20nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069456BDBM50069456(1-Methyl-1H-pyrrole-2-carboxylic acid (7-bromo-2,3...)
Affinity DataIC50: 20nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069461BDBM50069461(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 20nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069491BDBM50069491(1-(2-Methoxy-phenyl)-3-(7-nitro-2,3-dioxo-1,2,3,4-...)
Affinity DataIC50: 30nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069479BDBM50069479(5-Methyl-thiophene-2-carboxylic acid (7-bromo-2,3-...)
Affinity DataIC50: 30nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069470BDBM50069470(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 30nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069488BDBM50069488(1-(4-Methoxy-phenyl)-3-(7-nitro-2,3-dioxo-1,2,3,4-...)
Affinity DataIC50: 30nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069485BDBM50069485(2-Hydroxy-N-(7-nitro-2,3-dioxo-1,2,3,4-tetrahydro-...)
Affinity DataIC50: 40nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069464BDBM50069464(Furan-2-carboxylic acid (7-bromo-2,3-dioxo-1,2,3,4...)
Affinity DataIC50: 40nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069460BDBM50069460(N-(7-Nitro-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 40nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069490BDBM50069490(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 40nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069497BDBM50069497(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 40nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069467BDBM50069467(Acetic acid [(7-bromo-2,3-dioxo-1,2,3,4-tetrahydro...)
Affinity DataIC50: 40nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069481BDBM50069481(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 50nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069480BDBM50069480(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 50nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069475BDBM50069475(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 60nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069494BDBM50069494(N-(2,3-Dioxo-1,2,3,4-tetrahydro-quinoxalin-5-ylmet...)
Affinity DataIC50: 90nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069496BDBM50069496((7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin-5...)
Affinity DataIC50: 110nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069477BDBM50069477(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 110nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069466BDBM50069466(3,4,5-Trihydroxy-N-(7-nitro-2,3-dioxo-1,2,3,4-tetr...)
Affinity DataIC50: 150nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069476BDBM50069476(2-Amino-N-(7-nitro-2,3-dioxo-1,2,3,4-tetrahydro-qu...)
Affinity DataIC50: 170nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069469BDBM50069469(3,4,5-Trimethoxy-N-(7-nitro-2,3-dioxo-1,2,3,4-tetr...)
Affinity DataIC50: 200nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069484BDBM50069484(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 250nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069473BDBM50069473(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 280nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069487BDBM50069487(1-(7-Nitro-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 350nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069474BDBM50069474(N-(7-Nitro-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 630nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069463BDBM50069463(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 860nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069468BDBM50069468(1-(7-Nitro-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 900nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069462BDBM50069462(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069489BDBM50069489((7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin-5...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069493BDBM50069493(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069455BDBM50069455(2-Benzo[1,3]dioxol-5-yl-N-(7-bromo-2,3-dioxo-1,2,3...)
Affinity DataIC50: 3.90E+3nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069492BDBM50069492(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069472BDBM50069472(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069457BDBM50069457([2,3-Dioxo-8-(phenylacetylamino-methyl)-1,2,3,4-te...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Novartis Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069486BDBM50069486(N-(7-Bromo-2,3-dioxo-1,2,3,4-tetrahydro-quinoxalin...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro binding assay for the displacement of [3H]MDL-105519 from the glycine-site of NMDA receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed