Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 1174
TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM36363(CID6851947 | PAC-1 | US10166229, Example PAC-1)
Affinity DataEC50:  220nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM36364(CID9543559 | De-ally PAC-1 | US10166229, Example d...)
Affinity DataEC50:  430nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM36370(CID207112 | Piperazin-1-yl-acetic acid ethyl ester...)
Affinity DataEC50: >5.00E+4nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM36369(CID5060109 | (4-Benzylpiperazin-1-yl)-acetic acid ...)
Affinity DataEC50: >5.00E+4nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM50004308(1-Benzoylpiperazine | 1-Benzyl-piperazine, 10 | 1-...)
Affinity DataEC50: >5.00E+4nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM50125096(CHEMBL162522 | 1,4-Dibenzyl-piperazine, 9 | 1,4-Di...)
Affinity DataEC50: >5.00E+4nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM312057(US10166229, Example 00027)
Affinity DataEC50: >5.00E+4nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM36365(CID6885304 | (4-Benzylpiperazin-1-yl)-acetic acid ...)
Affinity DataEC50: >5.00E+4nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM36368(CID9543562 | (4-Benzylpiperazin-1-yl)-acetic acid ...)
Affinity DataEC50: >5.00E+4nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent

TargetCaspase-3(Human)
University of Illinois

US Patent
LigandPNGBDBM312058(US10166229, Example 00028)
Affinity DataEC50: >5.00E+4nMAssay Description:Procaspase-3 was recombinantly expressed in E. coli with an N-terminal His-6 tag (SEQ ID NO: 29) and purified. Immunoblotting was performed with an a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2019
Entry Details
US Patent