Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 8971
TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263478BDBM263478((s)-2-(6,8-dimethyl-4-oxobenzo[d][1,2,3]triazin-3(...)
Affinity DataKi:  1.00E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263499BDBM263499((s)-n-(1-(2-fluoro-4-(trifluoromethyl)phenyl)ethyl...)
Affinity DataKi:  1.10E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263493BDBM263493((s)-2-(5-methoxy-4-oxobenzo[d][1,2,3]triazin-3 (4h...)
Affinity DataKi:  2.60E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263461BDBM263461((s)-2-(6,8-dichloro-4-oxobenzo[d][1,2,3]triazin-3(...)
Affinity DataKi:  2.60E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263490BDBM263490((s)-2-(5-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  3.30E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263504BDBM263504((s)-n-(1-(2-fluoro-4-(trifluoromethoxy)phenyl)ethy...)
Affinity DataKi:  3.30E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263484BDBM263484((s)-n-(1-(2,4-dimethylphenyl)ethyl)-2-(6-fluoro-4-...)
Affinity DataKi:  3.90E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263487BDBM263487((s)-2-(6-fluoro-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  4.20E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263369BDBM263369((s)-2-(5-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  4.80E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263453BDBM263453((s)-2-(6-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  5.80E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263420BDBM263420((s)-n-(1-(2,4-dimethylphenyl)ethyl)-2-(4-oxobenzo[...)
Affinity DataKi:  6.30E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263459BDBM263459((s)-2-(8-methyl-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  7.20E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263486BDBM263486((s)-n-(1-(2-fluoro-4-methylphenyl)ethyl)-2-(6-fluo...)
Affinity DataKi:  7.70E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263482BDBM263482((s)-2-(8-fluoro-6-methyl-4-oxobenzo[d][1,2,3]triaz...)
Affinity DataKi:  8.50E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263474BDBM263474((s)-2-(5-methyl-4-oxobenzo[d][1,2,3]triazin-3 (4h)...)
Affinity DataKi:  9.20E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263503BDBM263503((s)-n-(1-(2-fluoro-4-(trifluoromethoxy)phenyl)ethy...)
Affinity DataKi:  9.30E+4nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263496BDBM263496((s)-2-(6-fluoro-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  1.06E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263457BDBM263457((s)-2-(8-chloro-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  1.10E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263492BDBM263492((s)-2-(6-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  1.15E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263509BDBM263509(n-(2-chloro-4-methoxyphenethyl)-2-(4-oxobenzo[d][1...)
Affinity DataKi:  1.17E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263368BDBM263368((s)-2-(4-oxobenzo[d][1,2,3]triazin-3(4h)-yl)-n-(1-...)
Affinity DataKi:  1.19E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263501BDBM263501((s)-n-(1-(4-(difluoromethoxy)phenyl)ethyl)-2-(5-me...)
Affinity DataKi:  1.20E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263502BDBM263502((s)-n-(1-(2-fluoro-4-(trifluoromethoxy)phenyl)ethy...)
Affinity DataKi:  1.20E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263489BDBM263489((s)-2-(6-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  1.28E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263440BDBM263440((s)-2-(4-oxobenzo[d][1,2,3]triazin-3(4h)-yl)-n-(1-...)
Affinity DataKi:  1.48E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263497BDBM263497((s)-n-(1-(2-fluoro-4-(trifluoromethyl)phenyl)ethyl...)
Affinity DataKi:  1.52E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263485BDBM263485((s)-n-(1-(2-fluoro-4-methylphenyl)ethyl)-2-(4-oxob...)
Affinity DataKi:  1.71E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263456BDBM263456((s)-2-(7-chloro-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  1.73E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263463BDBM263463((s)-2-(6-methyl-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  1.79E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263479BDBM263479((s)-2-(6,8-dimethyl-4-oxobenzo[d][1,2,3]triazin-3(...)
Affinity DataKi:  1.79E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263445BDBM263445((s)-2-(6-fluoro-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  1.82E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263511BDBM263511((s)-2-(4-oxobenzo[d][1,2,3]triazin-3(4h)-yl)-n-(1-...)
Affinity DataKi:  1.83E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263454BDBM263454((s)-2-(6-chloro-4-oxobenzo[d][1,2,3]triazin-3 (4h)...)
Affinity DataKi:  1.89E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263462BDBM263462((s)-2-(6,8-dichloro-4-oxobenzo[d][1,2,3]triazin-3(...)
Affinity DataKi:  1.90E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263512BDBM263512((s)-2-(4-oxobenzo[d][1,2,3]triazin-3 (4h)-yl)-n-(1...)
Affinity DataKi:  2.14E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263488BDBM263488((s)-2-(7-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  2.18E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263391BDBM263391((s)-n-(1-(4-chlorophenyl)ethyl)-2-(4-oxobenzo[d][1...)
Affinity DataKi:  2.28E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263494BDBM263494((s)-2-(8-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  2.40E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263500BDBM263500((s)-n-(1-(4-(difluoromethoxy)phenyl)ethyl)-2-(6-fl...)
Affinity DataKi:  2.82E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263469BDBM263469((s)-2-(7-methyl-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  3.47E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263495BDBM263495((s)-2-(8-methoxy-4-oxobenzo[d][1,2,3]triazin-3 (4h...)
Affinity DataKi:  3.52E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263491BDBM263491((s)-2-(7-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  3.75E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263480BDBM263480((s)-2-(4-oxo-6-(trifluoromethyl)benzo[d][1,2,3]tri...)
Affinity DataKi:  4.35E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263471BDBM263471((s)-2-(7-methoxy-4-oxobenzo[d][1,2,3]triazin-3(4h)...)
Affinity DataKi:  4.37E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263467BDBM263467((s)-2-(5-fluoro-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  4.59E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263370BDBM263370((s)-2-(4-oxobenzo[d][1,2,3]triazin-3(4h)-yl)-n-(1-...)
Affinity DataKi:  4.67E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263460BDBM263460((s)-n-(1-(4-methoxyphenyl)ethyl)-2-(8-methyl-4-oxo...)
Affinity DataKi:  5.26E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263477BDBM263477((s)-n-(1-(4-methoxyphenyl)ethyl)-2-(5-methyl-4-oxo...)
Affinity DataKi:  5.33E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263455BDBM263455((s)-2-(6-chloro-4-oxobenzo[d][1,2,3]triazin-3(4h)-...)
Affinity DataKi:  5.51E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

TargetProbable G-protein coupled receptor 139(Human)
Takeda Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 263473BDBM263473((s)-2-(5-methoxy-4-oxobenzo[d][1,2,3]triazin-3 (4h...)
Affinity DataKi:  6.19E+5nMAssay Description:This membrane based assay measures the ability of compounds to competitively bind GPR139 in stably transfected CHO-TRex membranes. CHO-TRex (Life Tec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2020
Entry Details
US Patent

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