Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 9463
TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 50529668BDBM50529668(Enobosarm | Gtx-024 | MK-2866 | Ostarine | US10806...)
Affinity DataIC50: 20nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 50529668BDBM50529668(Enobosarm | Gtx-024 | MK-2866 | Ostarine | US10806...)
Affinity DataKi:  20.2nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 50529647BDBM50529647(CHEMBL4584527 | US10806720, Compound 17 | US112305...)
Affinity DataKi:  28.4nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468351BDBM468351(US10806720, Compound 1036 | US11230523, Compound 1...)
Affinity DataIC50: 36.2nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468356BDBM468356(US10806720, Compound 1043 | US11648234, Compound 1...)
Affinity DataIC50: 57.9nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 50529667BDBM50529667(CHEMBL4444904 | US10806720, Compound 11 | US112305...)
Affinity DataIC50: 85.1nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468341BDBM468341(US10806720, Compound 1022)
Affinity DataIC50: 92.2nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 50529647BDBM50529647(CHEMBL4584527 | US10806720, Compound 17 | US112305...)
Affinity DataIC50: 95nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468362BDBM468362(US10806720, Compound 1058 | US11230523, Compound 1...)
Affinity DataIC50: 132nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468326BDBM468326(US10806720, Compound 1006 | US11230523, Compound 1...)
Affinity DataIC50: 149nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468324BDBM468324(US10806720, Compound 1004 | US11230523, Compound 1...)
Affinity DataIC50: 179nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468339BDBM468339(US10806720, Compound 1020 | US11648234, Compound 1...)
Affinity DataIC50: 192nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468304BDBM468304(US10806720, Compound 100 | US11230523, Compound 10...)
Affinity DataKi:  198nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468322BDBM468322(US10806720, Compound 1002 | US11648234, Compound 1...)
Affinity DataIC50: 199nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468333BDBM468333(US10806720, Compound 1014 | US11230523, Compound 1...)
Affinity DataIC50: 205nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 50425732BDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 216nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468364BDBM468364(US10806720, Compound 1063 | US11230523, Compound 1...)
Affinity DataIC50: 217nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468331BDBM468331(US10806720, Compound 1012 | US11230523, Compound 1...)
Affinity DataIC50: 219nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468329BDBM468329(US10806720, Compound 1010 | US11230523, Compound 1...)
Affinity DataIC50: 226nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468345BDBM468345(US10806720, Compound 1028 | US11230523, Compound 1...)
Affinity DataKi:  227nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 18678BDBM18678(CHEMBL63560 | (2R)-N-[4-cyano-3-(trifluoromethyl)p...)
Affinity DataIC50: 248nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468358BDBM468358(US10806720, Compound 1045 | US11648234, Compound 1...)
Affinity DataIC50: 251nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468329BDBM468329(US10806720, Compound 1010 | US11230523, Compound 1...)
Affinity DataKi:  259nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 50529667BDBM50529667(CHEMBL4444904 | US10806720, Compound 11 | US112305...)
Affinity DataKi:  267nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468363BDBM468363(US10806720, Compound 1059 | US11230523, Compound 1...)
Affinity DataIC50: 285nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468357BDBM468357(US10806720, Compound 1044 | US11648234, Compound 1...)
Affinity DataIC50: 317nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468324BDBM468324(US10806720, Compound 1004 | US11230523, Compound 1...)
Affinity DataKi:  322nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468321BDBM468321(US10806720, Compound 1001 | US11230523, Compound 1...)
Affinity DataKi:  328nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468352BDBM468352(US10806720, Compound 1037 | US11230523, Compound 1...)
Affinity DataIC50: 350nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468336BDBM468336(US10806720, Compound 1017 | US11230523, Compound 1...)
Affinity DataIC50: 404nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468359BDBM468359(US10806720, Compound 1050 | US11230523, Compound 1...)
Affinity DataIC50: 427nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468342BDBM468342(US10806720, Compound 1024 | US11648234, Compound 1...)
Affinity DataIC50: 464nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 18678BDBM18678(CHEMBL63560 | (2R)-N-[4-cyano-3-(trifluoromethyl)p...)
Affinity DataKi:  509nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468333BDBM468333(US10806720, Compound 1014 | US11230523, Compound 1...)
Affinity DataKi:  512nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468304BDBM468304(US10806720, Compound 100 | US11230523, Compound 10...)
Affinity DataIC50: 531nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468363BDBM468363(US10806720, Compound 1059 | US11230523, Compound 1...)
Affinity DataKi:  601nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468362BDBM468362(US10806720, Compound 1058 | US11230523, Compound 1...)
Affinity DataKi:  606nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468343BDBM468343(US10806720, Compound 1025 | US11230523, Compound 1...)
Affinity DataKi:  612nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468340BDBM468340(US10806720, Compound 1021 | US11230523, Compound 1...)
Affinity DataKi:  633nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468350BDBM468350(US10806720, Compound 1035 | US11648234, Compound 1...)
Affinity DataIC50: 758nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468331BDBM468331(US10806720, Compound 1012 | US11230523, Compound 1...)
Affinity DataKi:  821nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468349BDBM468349(US10806720, Compound 1034 | US11648234, Compound 1...)
Affinity DataIC50: 827nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468336BDBM468336(US10806720, Compound 1017 | US11230523, Compound 1...)
Affinity DataKi:  898nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468348BDBM468348(US10806720, Compound 1032 | US11648234, Compound 1...)
Affinity DataIC50: 901nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468326BDBM468326(US10806720, Compound 1006 | US11230523, Compound 1...)
Affinity DataKi:  906nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468327BDBM468327(US10806720, Compound 1007 | US11648234, Compound 1...)
Affinity DataIC50: 959nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468343BDBM468343(US10806720, Compound 1025 | US11230523, Compound 1...)
Affinity DataIC50: 969nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468338BDBM468338(US10806720, Compound 1019 | US11648234, Compound 1...)
Affinity DataIC50: 1.01E+3nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468335BDBM468335(US10806720, Compound 1016 | US11230523, Compound 1...)
Affinity DataIC50: 1.02E+3nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

TargetAndrogen receptor(Human)
University of Tennessee Research Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 468325BDBM468325(US10806720, Compound 1005 | US11648234, Compound 1...)
Affinity DataIC50: 1.02E+3nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2021
Entry Details
US Patent

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