Compile Data Set for Download or QSAR
Report error Found 623 Enz. Inhib. hit(s) with all data for entry = 9905
TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497971BDBM497971(US11008314, Compound 59)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498037BDBM498037(US11008314, Compound 121)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498036BDBM498036(US11008314, Compound 120)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase JAK3(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498035BDBM498035(US11008314, Compound 119)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498035BDBM498035(US11008314, Compound 119)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498035BDBM498035(US11008314, Compound 119)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498034BDBM498034(US11008314, Compound 118)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase JAK3(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498034BDBM498034(US11008314, Compound 118)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498034BDBM498034(US11008314, Compound 118)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497967BDBM497967(US11008314, Compound 56)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase JAK3(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498041BDBM498041(US11008314, Compound 125)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498041BDBM498041(US11008314, Compound 125)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498041BDBM498041(US11008314, Compound 125)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498040BDBM498040(US11008314, Compound 124)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase JAK3(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498040BDBM498040(US11008314, Compound 124)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498040BDBM498040(US11008314, Compound 124)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497974BDBM497974(US11008314, Compound 62)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498040BDBM498040(US11008314, Compound 124)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498039BDBM498039(US11008314, Compound 123)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498038BDBM498038(US11008314, Compound 122)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497907BDBM497907(US11008314, Compound 1)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498045BDBM498045(US11008314, Compound 129)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497907BDBM497907(US11008314, Compound 1)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497978BDBM497978(US11008314, Compound 66)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498042BDBM498042(US11008314, Compound 126)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498050BDBM498050(US11008314, Compound 133)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498050BDBM498050(US11008314, Compound 133)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497912BDBM497912(US11008314, Compound 7)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498048BDBM498048(US11008314, Compound 132)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497910BDBM497910(US11008314, Compound 5)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498047BDBM498047(US11008314, Compound 131)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497910BDBM497910(US11008314, Compound 5)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498046BDBM498046(US11008314, Compound 130)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498054BDBM498054(US11008314, Compound 137)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498054BDBM498054(US11008314, Compound 137)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498054BDBM498054(US11008314, Compound 137)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497918BDBM497918(US11008314, Compound 11)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497987BDBM497987(US11008314, Compound 75)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498053BDBM498053(US11008314, Compound 136)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498010BDBM498010(US11008314, Compound 135 | US11008314, Compound 98)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498010BDBM498010(US11008314, Compound 135 | US11008314, Compound 98)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497986BDBM497986(US11008314, Compound 74)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498010BDBM498010(US11008314, Compound 135 | US11008314, Compound 98)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497916BDBM497916(US11008314, Compound 9)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498051BDBM498051(US11008314, Compound 134)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase TXK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498051BDBM498051(US11008314, Compound 134)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497985BDBM497985(US11008314, Compound 73)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 498051BDBM498051(US11008314, Compound 134)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497915BDBM497915(US11008314, Compound 8)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Corvus Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 497923BDBM497923(US11008314, Compound 15)
Affinity DataIC50: 10nMAssay Description:The potency of inhibition is measured by binding affinity.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2021
Entry Details
US Patent

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