Compile Data Set for Download or QSAR
maximum 50k data
Found 592 Enz. Inhib. hit(s) with all data for entry = 10710
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561275((6-(4-((4-(1H- pyrazol-4-yl) phenyl)amino)-6,7- di...)
Affinity DataIC50:  4nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561220(6-(4-((1H- indazol-5- yl)amino)- pyrimidin-2- yl)-...)
Affinity DataIC50:  5nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561252((3,3- difluoroazetidin- 1-yl)(6-(4-((3- methoxy-4-...)
Affinity DataIC50:  6nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561112(6-(4-((4-(1H-pyrazol-4- yl)phenyl)amino)pyrimidin-...)
Affinity DataIC50:  6nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561244(6-(4-((4-(1H- pyrazol-4- yl)phenyl)- amino)- pyrim...)
Affinity DataIC50:  8nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561249((3,3- difluoroazetidin- 1-yl)(6-(4-((3- fluoro-4- ...)
Affinity DataIC50:  9nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561242(6-(4-((4-(1H- pyrazol-4- yl)phenyl)- amino)- pyrim...)
Affinity DataIC50:  9nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561294((5-(4-((4-(1H-pyrazol- 4-yl)phenyl)amino)-6,7- dih...)
Affinity DataIC50:  10nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561274((6-(4-((4-(1H- pyrazol-4-yl) phenyl)amino)-5,7- di...)
Affinity DataIC50:  10nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561115((6-(4-((4-(1H-pyrazol-4- yl)phenyl)amino)pyrimidin...)
Affinity DataIC50:  11nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561221(6-(4-((1H- indazol-5- yl)amino)- pyrimidin-2- yl)-...)
Affinity DataIC50:  11nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561262((6-(4-((4-1H- pyrazol-4-yl) phenyl)amino)-5- fluor...)
Affinity DataIC50:  12nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM402404(US10329282, Compound TDI01433 | US11390609, Compou...)
Affinity DataIC50:  13nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561132(1-(6-(4-((4- (1H-pyrazol-4- yl)phenyl)- amino)- py...)
Affinity DataIC50:  13nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561108(1-(6-(4-((4-(1H-pyrazol-4- yl)phenyl)amino)pyrimid...)
Affinity DataIC50:  13nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561225(6-(4-((1H- indazol-5- yl)amino)- pyrimidin-2- yl)-...)
Affinity DataIC50:  14nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561276((6-(4-((4-(1H- pyrazol-4-yl) phenyl)amino)-6- meth...)
Affinity DataIC50:  14nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561230((6-(4-((4-(1H- pyrazol-4- yl)phenyl)amino)- 6,7-di...)
Affinity DataIC50:  15nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561146((6-(4-((4-(1H-pyrazol-4-yl)phenyl) amino)pyrimidin...)
Affinity DataIC50:  15nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561111(6-(4-((4-(1H- pyrazol-4- yl)phenyl)- amino)- pyrim...)
Affinity DataIC50:  15nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561196(2- azaspiro[3.3]heptan 6-yl 5-(4-((4-(1H- pyrazol-...)
Affinity DataIC50:  16nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM402391(US10329282, Compound TDI01398 | US11390609, Compou...)
Affinity DataIC50:  16nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM402322(US10329282, Compound TDI01153 | US11390609, Compou...)
Affinity DataIC50:  16nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561289((5-(4-((4-(1H-pyrazol-4- yl)phenyl)amino)furo[3,2-...)
Affinity DataIC50:  18nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561213(6-(4-((1H- indazol-5- yl)amino)- pyrimidin-2- yl)-...)
Affinity DataIC50:  18nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561123((6-(4-((4-(1H-pyrazol-4- yl)phenyl)amino)pyrimidin...)
Affinity DataIC50:  18nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM402367(US10329282, Compound TDI01318 | US11390609, Compou...)
Affinity DataIC50:  18nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561070(6-(4-((1H- indazol-5- yl)amino)- pyrimidin-2- yl)-...)
Affinity DataIC50:  18nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561255((6-(4-((4-(1H- pyrazol-4-yl) phenyl)amino)-5- meth...)
Affinity DataIC50:  18nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561174(3,3- difluorocyclobutyl 5-(4-((1H-indazol-5- yl)am...)
Affinity DataIC50:  19nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561272((6-(4-((4-(1H- pyrazol-4-yl) phenyl)amino)-5- meth...)
Affinity DataIC50:  19nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561157((3,3- difluorocyclobutyl)(5- (4-((2-methoxy-4-(1H-...)
Affinity DataIC50:  21nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561171((5-(4-((4-(1H-pyrazol-4- yl)phenyl)amino)pyrimidin...)
Affinity DataIC50:  22nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561138((6-(4-((4-(1H-pyrazol-4-yl) phenyl)amino)pyrimidin...)
Affinity DataIC50:  22nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM402298(US10329282, Compound TDI01108 | US11390609, Compou...)
Affinity DataIC50:  22nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561165(3,3- difluorocyclobutyl 5-(4-((4-(1H- pyrazol-4- y...)
Affinity DataIC50:  23nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM402339(US10329282, Compound TDI01200 | US11390609, Compou...)
Affinity DataIC50:  23nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561254((6-(4-((4-(1H- pyrazol-4- yl)phenyl)amino)-5- meth...)
Affinity DataIC50:  23nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561176((6-(4-((4-(1H- pyrazol-4- yl)phenyl)amino)-5- fluo...)
Affinity DataIC50:  24nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM402323(US10329282, Compound TDI01156 | US11390609, Compou...)
Affinity DataIC50:  25nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561180(1-(4-((4-(1H-pyrazol-4- yl)phenyl)amino)-2-(2- (3,...)
Affinity DataIC50:  25nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561155(US11390609, Compound TDI01546)
Affinity DataIC50:  26nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561055((6-(4-((1H- indazol-5- yl)amino)- pyrimidin- 2-yl)...)
Affinity DataIC50:  26nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561245(6-(4-((4-(1H- pyrazol-4- yl)phenyl)- amino)- pyrim...)
Affinity DataIC50:  26nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM402411(US10329282, Compound TDI01847B | US11390609, Compo...)
Affinity DataIC50:  26nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561273(5-(4-((4-(1H- pyrazol-4- yl)phenyl)amino) pyrimidi...)
Affinity DataIC50:  27nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561188(3,3- difluorocyclobutyl 5-(4-((1H-indazol-5- yl)am...)
Affinity DataIC50:  27nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561263((6-(4-((6-(1H- pyrazol-4-yl) pyridin-3- yl)amino) ...)
Affinity DataIC50:  27nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561251(N-(3-fluoro-4- (1H-pyrazol-4- yl)phenyl)-2- (2-(th...)
Affinity DataIC50:  27nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRho-associated protein kinase 2(Homo sapiens (Human))
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM561195((6-(4-((4-(1H- pyrazol-4-yl) phenyl)amino)-6,7- di...)
Affinity DataIC50:  27nMAssay Description:The kinase IC50 was determined by a commercialized CISBIO kinase detection kit, HTRF KinEASE-STK S2 kit (62ST2PEC). ROCK2 (01-119) employed in the re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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