Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 8230
TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 1.90nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 5.10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791820BDBM791820(US12545652, Comparative Compound A)
Affinity DataIC50: 10nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK1(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 20nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK1(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 26nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK1(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791820BDBM791820(US12545652, Comparative Compound A)
Affinity DataIC50: 49nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK2(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 50nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK2(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 77nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK2(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791820BDBM791820(US12545652, Comparative Compound A)
Affinity DataIC50: 87nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK3(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 212nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK3(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 271nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetTyrosine-protein kinase JAK3(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791820BDBM791820(US12545652, Comparative Compound A)
Affinity DataIC50: 290nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2C9(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 4.40E+3nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2C8(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 8.20E+3nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2C9(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 2.60E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2C19(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2D6(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 3A4(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 1A2(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2B6(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2C8(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2C19(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2D6(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 3A4(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791822BDBM791822(US12545652, Compound (1))
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 1A2(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent

TargetCytochrome P450 2B6(Human)
Sareum

US Patent
LigandChemical structure of BindingDB Monomer ID 791821BDBM791821(US12545652, Comparative Compound B)
Affinity DataIC50: 3.00E+4nMAssay Description:NMDA receptors are ion channels that are highly permeable to Ca2+ ions, rendering it possible to monitor NMDA receptor function using cell-based calc...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/22/2026
Entry Details ArticleUS Patent